No known drug interactions for the matched ingredients — not a guarantee none exist. Check your meds →
Dietary supplement

Betaine Unflavored Ingredients & Drug Interactions

by Axe & Sledge Supplements

Powder Category: Non-nutrient/non-botanical
No known interaction
The interaction bottom line No known interaction

Betaine Unflavored is a dietary supplement by Axe & Sledge Supplements with 1 active ingredient. Its ingredients are commonly taken for high homocysteine levels, liver health (fatty liver), exercise performance and strength.We don’t currently list a known drug interaction for its mapped ingredients — but that doesn’t guarantee none exist, so always confirm with your pharmacist.

HelloPharmacist Scorecard of Betaine Unflavored by Axe & Sledge Supplements

Our pharmacy team’s full take, with four database checks built into the cards below — a summary of what is known, not a grade of the product itself.

From our pharmacy team — supplement deep dive

What’s inside

Full disclosure
Ingredient Transparency · database check
Full

Every active ingredient lists its own amount on the label.

Why this rating?
  • The label discloses an exact amount for 1 of its 1 active ingredient.
  • No proprietary blends here — you can verify the dose of every single component.

This product contains a single active ingredient: betaine anhydrous. Betaine is a naturally occurring compound that plays a role in how your body handles a substance called homocysteine — an amino acid your cells produce during normal metabolism.

The powder form lets you mix it into drinks or food as needed.

Does it work?

Strong evidence
Evidence for Intended Use · database check
By FDA rules, dietary supplements can’t claim to treat, cure, or prevent disease — so labels speak in careful marketing language. We discern each product’s intended use from its name, label claims, and label statements, then grade the clinical evidence for that use. How these ratings are computed
Strong

Clinical evidence supports at least one of this product's ingredients for its stated purpose.

Why this rating?
  • The label markets this product for: supports cardiovascular health and homocysteine levels.
  • We looked for evidence on: Hyperhomocysteinemia, Homocystinuria, Nonalcoholic steatohepatitis (NASH), Hepatitis C, Metabolic Syndrome, blood vessel function — and 1 related terms.
  • The strongest evidence on file: Betaine Anhydrous is rated "Effective" for Homocystinuria (Natural Medicines).
  • Also on file: Betaine Anhydrous is rated "Possibly Effective" for Hyperhomocysteinemia.
  • Also on file: Betaine Anhydrous is rated "Insufficient Reliable Evidence To Rate" for Hepatitis C, Nonalcoholic steatohepatitis (NASH), Metabolic Syndrome.

Betaine anhydrous is effective for homocystinuria, a genetic condition where homocysteine builds up to harmful levels in the blood. It's possibly effective for hyperhomocysteinemia, a milder elevation of homocysteine linked to heart health.

For nonalcoholic fatty liver disease (NASH), depression, and reflux disease (GERD), the evidence isn't established well enough for us to rate it — meaning we don't have enough reliable data to say whether it works for those uses.

The evidence, ingredient by ingredient Betaine Anhydrous

How safe is it?

Well-documented data
Safety Information · database check
Well characterized

Adverse-effect, pregnancy, and general safety data are on file for most of these ingredients.

Why this rating?
  • We hold adverse-effect (side-effect) data for 1 of the 1 matched ingredient.
  • Pregnancy & breastfeeding safety ratings cover 1 of 1.
  • General safety write-ups exist for 1 of 1.
  • Remember: this measures how much safety information exists. Thin data is not the same as being safe.

Betaine anhydrous is generally well tolerated at studied doses, but the safety data overall isn't robust. The most common side effects are body odor, diarrhea, nausea, vomiting, and GI distress — mostly mild and manageable.

Rarely, cerebral edema (fluid buildup in the brain) has been reported, though this is uncommon. Safety during breastfeeding is not well established, so if you're nursing, talk with your doctor or pharmacist before starting.

There isn't enough reliable safety data in pregnancy either — your healthcare provider is the right person to discuss that with before use.

Side effects, ingredient by ingredient Betaine Anhydrous

Meds to double-check

No known interactions
Known Interaction Concern · database check
No known interactions

No medication interactions are currently documented for the matched ingredients — that isn't a guarantee none exist.

Why this rating?
  • None of the 1 matched ingredient has a documented medication interaction on file.

No interactions are documented in our data for betaine anhydrous. That doesn't mean none exist — it just means we have no information in our files showing it affects how specific drugs work.

Run your exact medications through the checker on this page to be thorough.

The bottom line

Scorecard at a glanceFully disclosed formula with clinical evidence supporting its stated purpose. No medication interactions are currently documented, and safety information is well characterized.

Betaine anhydrous is a good fit if you have homocystinuria or your doctor has told you your homocysteine is elevated and has recommended betaine. If you're considering it for other reasons — like fatty liver disease, mood, or reflux — talk with your pharmacist or doctor first, since the evidence isn't clear.

Check with your healthcare provider before starting, especially if you're pregnant or breastfeeding.

Educational only — not medical advice; always confirm with your pharmacist. Our editorial policy · How we use AI

Assessment coverage: 1 of 1 active ingredient matched to our full ingredient reviews (monographs). Based on the product label dated Sep 24, 2021.

This Scorecard evaluates available label information, ingredient evidence, and known medication-safety considerations. It does not independently verify product identity, purity, potency, contamination, or manufacturing quality. How these ratings are computed

At a glance

General information

Key facts about Betaine Unflavored, straight from the product label.

Brand Axe & Sledge Supplements
Barcode (UPC) 750258225969
Net contents 100 Gram(s); 3.53 Ounce(s)
Market status On market
Date entered into DSLD Sep 24, 2021
DSLD ID 254854
Product type Non-nutrient/non-botanical
Supplement form Powder
Dietary claims / uses All Other, Structure/Function
Intended target group(s) Adult (18 - 50 Years), Women (not pregnant or lactating)
From the label
Everything in this section is reproduced from the manufacturer’s own product label — it’s the label speaking, not HelloPharmacist. We show it so you can see exactly what the maker states; we don’t verify or endorse those statements.

Supplement Facts

The label details for Betaine Unflavored by Axe & Sledge Supplements, sourced from the NIH Dietary Supplement Label Database.

Supplement Facts

Daily Value (DV) Target Group(s):
Adults and children 4 or more years of age
Minimum serving Sizes:
2.5 Gram(s)
Maximum serving Sizes:
2.5 Gram(s)
Servings per container
40
UPC/BARCODE
750258225969
IngredientAmount% DV
Betaine Anhydrous2500 mg--

Other ingredients: None

Tap any ingredient to jump to its full detail below.

Label statements
These statements are the manufacturer’s wording, reproduced from the product label — the label is saying it, not HelloPharmacist. We don’t verify or endorse them.
Suggested/Recommended/Usage/Directions

Suggested use As a dietary supplement, mix 2.5 grams with 6 to 8 oz. of water or your favorite beverage. Best if taken prior to workout. Do not exceed 1 serving per day.

General Statements

For the hardest workers in the gym

Axe and Sledge basics

Precautions

Warning: Consult with a physician prior to use if you have a medical condition.

Don't use if pregnant or lactating.

Keep out of reach of children.

Storage

Keep container tightly closed in a cool, dry and dark place.

FDA Disclaimer Statement

These statements have not been evaluated by the Food and Drug Administration. This product is not intended to diagnose, treat, cure, or prevent any disease.

Formulation

Supports a healthy cardiovascular system Supports healthy homocysteine levels Supports healthy blood vessel and liver function

Contains no fillers, excipients or artificial substances.

FDA Statement of Identity

Dietary Supplement

See for yourself

Betaine Unflavored by Axe & Sledge Supplements label

The label scan from the NIH Dietary Supplement Label Database. Tap to enlarge.

What’s inside

The Ingredients in Betaine Unflavored by Axe & Sledge Supplements

This is the 1 active ingredient this product is made of. Select it to open its full monograph.

Serving size2.5 Gram(s) Dosage formPowder Servings per container40 Amounts shown are per serving.

Betaine Anhydrous

No known
interactions
2500 mg per serving

Betaine anhydrous (also called trimethylglycine) is a compound found in foods like beets, spinach, and whole grains, and is sold as a supplement and a...

Betaine Anhydrous monograph & interactions

Other (inactive) ingredients: None. These complete the product’s ingredient list but are not active constituents.

Interaction report

Betaine Unflavored by Axe & Sledge Supplements Drug Interactions

We don’t currently list any known drug interactions for the mapped ingredients in Betaine Unflavored. This doesn’t guarantee none exist — always confirm with your pharmacist before combining a supplement with your medications.

The maker

Brand information

Manufacturer and brand details for Betaine Unflavored, from the product label.

Axe & Sledge Supplements

See all Axe & Sledge Supplements products
Name
Axe & Sledge Supplements
Street Address
1909 New Texas Road
City
Pittsburgh
State
PA
ZipCode
15239
Phone Number
(888) 944-6612
Web Address
www.axeandsledge.com
Pharmacist Counseling Corner

Betaine Unflavored by Axe & Sledge Supplements: Common Questions

Does Betaine Unflavored by Axe & Sledge Supplements interact with any medications?
We do not currently list a known interaction for the mapped ingredients in Betaine Unflavored. This does not guarantee none exist, so confirm with your pharmacist.
How can one product interact with so many drugs?
Betaine Unflavored contains a single active ingredient, and that one ingredient can interact with many different medications on its own. We check it against each medication and show the mechanism responsible.
Where does this information come from?
The product label data comes from the NIH Dietary Supplement Label Database (DSLD); the interaction data is built on the Natural Medicines database and reviewed by HelloPharmacist pharmacists.
What does betaine anhydrous actually do in my body?
Betaine helps your body manage homocysteine, an amino acid your cells produce naturally. High levels of homocysteine can be a problem for your heart and blood vessels, and betaine helps bring those levels down.
Will this give me bad body odor?
Body odor is the most commonly reported side effect in the studies. It's not guaranteed to happen, but it's something to be aware of. If it does occur, talking with your pharmacist about dose adjustments might help.
Can I take this if I'm breastfeeding?
Safety while breastfeeding isn't well established, so caution is advised. Talk with your doctor or pharmacist before starting — they can weigh whether the benefit outweighs the unknowns for your specific situation.
Is this powder pure betaine, or does it have fillers?
According to the product facts, there are no inactive ingredients listed — it's just the betaine anhydrous powder.
Does betaine work for fatty liver disease?
There isn't enough reliable evidence yet to say whether betaine helps with nonalcoholic fatty liver disease. Your doctor can advise whether it's worth trying in your case.

Written and reviewed by the HelloPharmacist editorial staff. Our editorial policy

Not sure if Betaine Unflavored is safe with your meds?

Our pharmacists answer your medication & supplement questions — free.

Ask a pharmacist

Label information is sourced from the NIH Dietary Supplement Label Database and reflects the product version on file; always read your actual product label. This page is for education only and is not a substitute for professional medical advice. Confirm with your pharmacist or doctor before combining supplements and medications.

Betaine Unflavored label
Go deeper

The Full Monographs Behind Betaine Unflavored’s Ingredients

Every ingredient we hold a full HelloPharmacist monograph for — uses, evidence, safety, and the complete interaction list.

Sources

Sources & How We Checked

Betaine Unflavored's label data comes from the NIH Dietary Supplement Label Database; the ingredient interaction data is from the Natural Medicines database, reviewed by our pharmacists.

Content is written and reviewed by licensed HelloPharmacist pharmacists. See our data sources and editorial standards for how this information is built and checked.

The 11 references behind this product’s interaction data

Every citation that drives the interaction findings for this product’s ingredients, from the evidence-graded Natural Medicines (TRC Healthcare) database. Open an ingredient to browse its citations — links open the study on PubMed or the publisher’s site.

Betaine Anhydrous 11 references
  1. Cystadane (betaine anhydrous for oral solution) Package insert. Orphan Medical, Inc. Minnetonka, MN. November 2005.
  2. Abdelmalek MF, Angulo P, Jorgensen RA, et al. Betaine, a promising new agent for patients with nonalcoholic steatohepatitis: results of a pilot study. Am J Gastroenterol 2001;96:2711-7.. PubMed
  3. Schwab U, Torronen A, Toppinen L, et al. Betaine supplementation decreases plasma homocysteine concentrations but does not affect body weight, body composition, or resting energy expenditure in human subjects. Am J Clin Nutr 2002;76:961-7. PubMed
  4. McGregor DO, Dellow WJ, Robson RA, et al. Betaine supplementation decreases post-methionine hyperhomocysteinemia in chronic renal failure. Kidney Int 2002;61:1040-6. PubMed
  5. Olthof MR, van Vliet T, Verhoef P, et al. Effect of homocysteine-lowering nutrients on blood lipids: results from four randomised, placebo-controlled studies in healthy humans. PloS Med 2005;2:e135. PubMed
  6. Knopman, D. and Patterson, M. An open-label, 24-week pilot study of the methyl donor betaine in Alzheimer disease patients. Alzheimer Dis.Assoc.Disord. 2001;15(3):162-165. PubMed
  7. Moat, S. J., Madhavan, A., Taylor, S. Y., Payne, N., Allen, R. H., Stabler, S. P., Goodfellow, J., McDowell, I. F., Lewis, M. J., and Lang, D. High- but not low-dose folic acid improves endothelial function in coronary artery disease. Eur J Clin Invest 2 PubMed
  8. Abdelmalek, M. F., Sanderson, S. O., Angulo, P., Soldevila-Pico, C., Liu, C., Peter, J., Keach, J., Cave, M., Chen, T., McClain, C. J., and Lindor, K. D. Betaine for nonalcoholic fatty liver disease: results of a randomized placebo-controlled trial. Hepa PubMed
  9. Ashtary-Larky D, Bagheri R, Ghanavati M, et al. Effects of betaine supplementation on cardiovascular markers: a systematic review and meta-analysis. Crit Rev Food Sci Nutr. 2021 Mar 25:1-18. PubMed
  10. Zawieja EE, Zawieja B, Chmurzynska A. Betaine supplementation moderately increases total cholesterol levels: a systematic review and meta-analysis. J Diet Suppl. 2021;18(1):105-117. PubMed
  11. Imbard A, Toumazi A, Magréault S, et al. Efficacy and pharmacokinetics of betaine in CBS and cblC deficiencies: a cross-over randomized controlled trial. Orphanet J Rare Dis 2022;17(1):417. PubMed

See these in context on the Betaine Anhydrous monograph →

Parts of this content are provided by the Therapeutic Research Center, LLC.

DISCLAIMER: Currently this does not check for drug-drug interactions. This is not an all-inclusive comprehensive list of potential interactions and is for informational purposes only. Not all interactions are known or well-reported in the scientific literature, and new interactions are continually being reported. Input is needed from a qualified healthcare provider including a pharmacist before starting any therapy. Application of clinical judgment is necessary.

© 2021 Therapeutic Research Center, LLC

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