FDA-filed SPL labeling · retrieved through openFDA

Acyclovir / Hydrocortisone

Acyclovir/hydrocortisone is a combination antiviral and anti-inflammatory cream used to treat recurrent herpes labialis (cold sores) on the lips and around the mouth.

Brand name Xerese
Drug classes Herpes Simplex Virus Nucleoside Analog Dna Polymerase Inhibitor
Rx Form 1 Route Topical
Dr. Brian Staiger, PharmD, BCPS
Reviewed by Last reviewed Aug 3, 2026
🧬 Where this information comes from Click to expand

The clinical label records used on this page are FDA-filed Structured Product Labeling (SPL) retrieved through openFDA. We identified 1 clinical label set within the page’s selected clinical scope after exact ingredient or ingredient-combination matching and applicable route/form matching. Forms, routes, brands, labelers, strengths, and NDC product-record counts are built separately from matching FDA National Drug Code Directory records. The linked DailyMed document is a representative official source for verification, not the page’s only clinical source. View the linked label on DailyMed →

At a glance
Linked label effectiveAug 3, 2020
AvailabilityRx
Earliest approval/marketing year 2009
FDA-listed product records 1
Boxed warningNone found in compared labels
How we combine label and product data →
No current FDA shortage listed · checked Sep 17, 2026
Acyclovir / Hydrocortisone at a glance The quick version — the full detail is in the Patient Information Guide below.
💊
HelloPharmacist Editorial Team Bottom Line
Xerese cream combines an antiviral (acyclovir) and a mild anti-inflammatory (hydrocortisone) to treat recurrent cold sores on the lips and surrounding skin in adults and children 6 and older. Start it at the very first sign of a cold sore and apply it five times a day for five days. If a sore isn't healing within two weeks, check with your doctor — not all lip lesions are cold sores.

📖 Acyclovir / Hydrocortisone: Patient Information Guide

A plain-language walkthrough of Acyclovir / Hydrocortisone — what it treats, how it works, how it’s taken, side effects, warnings and interactions. Tap any section to expand it.

🎯What it's used for

Acyclovir/hydrocortisone is a topical combination medication supported for the following use:

  • Xerese cream is indicated for the early treatment of recurrent herpes labialis (cold sores) on the lips and skin around the mouth in adults and children 6 years of age and older.
  • Xerese is used to reduce the likelihood that a cold sore will become an ulcerative (open) sore.
  • Xerese is used to shorten the time it takes a cold sore lesion to heal.
⚙️How it works

Acyclovir is an antiviral drug that works by mimicking the building blocks of viral DNA. Herpes simplex virus (HSV-1 and HSV-2) activates acyclovir inside infected cells by converting it into an active form that blocks the viral enzyme needed to copy the virus's genetic material. This stops the virus from replicating and spreading. Hydrocortisone is a mild corticosteroid that reduces the inflammation — swelling, redness, and irritation — associated with a cold sore outbreak.

One thing worth knowing: like other antiviral drugs, acyclovir can lose effectiveness if the virus develops resistance — a change in the viral enzymes that makes the drug less able to block replication. This is more of a concern in people with weakened immune systems or those who experience repeated treatment failures.

💊How it's taken

Xerese cream is applied to the affected area five times a day for five days. Starting treatment early — at the very first tingle, itch, or redness — gives the best results. Apply a thin layer that covers the sore and its surrounding edge.

  • Use it five times per day for exactly five days.
  • Apply as soon as the first symptoms appear — early use matters.
  • Avoid rubbing the area more than needed; it can aggravate or spread the infection.
  • This is for skin use only — not for internal use. Follow your prescriber and the label for all details.
🤒Side effects — in detail

The most commonly reported side effects with Xerese are local skin reactions at the application site:

  • Skin irritation where the cream is applied
  • Contact sensitization — an allergic-type skin reaction at the site
  • Skin dryness or flaking

If you notice a sore that isn't healing within two weeks, or if your skin reaction seems severe or is spreading, contact your doctor — this could point to a different type of infection or an allergic reaction that needs attention.

⚠️Warnings & precautions
  • For external use only: Xerese should only be applied to the lips and surrounding skin. Never use it in or near the eye, inside the mouth or nose, or on the genitals.
  • Not all lip sores are cold sores: Bacterial and fungal infections can look similar to herpes labialis. If the sore doesn't start to heal within 2 weeks, see a doctor.
  • Skin irritation and allergic reactions: Xerese can cause irritation or contact sensitization at the site. If you notice worsening redness, swelling, or a rash, stop using it and contact your doctor.
  • Immunocompromised patients: People with weakened immune systems (such as those with HIV) should talk to their doctor before using Xerese — the benefit in this group has not been adequately established.
  • Corticosteroid absorption: Although absorption through the skin is expected to be low when used as directed, broken or inflamed skin can allow more hydrocortisone to enter the bloodstream.
🔀What it interacts with

No formal drug interaction studies have been conducted with Xerese. Talk to your pharmacist or doctor about all medications, supplements, and skin products you use alongside Xerese.

  • Other topical products: Using other creams or ointments on the same area at the same time has not been studied — check with your doctor before combining treatments.

This is not a complete list of interactions. Always talk with your doctor or pharmacist before starting, stopping, or changing any medication.

📋Before taking it
  • Children under 6: Safety and effectiveness of Xerese have not been established in children younger than 6 years of age.
  • Pregnancy: Tell your doctor if you are pregnant. Published observational data on topical acyclovir and low-potency topical corticosteroids have not shown a clear association with birth defects or pregnancy complications, and systemic absorption from topical Xerese is expected to be minimal — but discuss any concerns with your doctor.
  • Breastfeeding: There are no data on whether acyclovir or hydrocortisone pass into breast milk after topical application. Discuss use of Xerese with your doctor if you are breastfeeding.
  • Weakened immune system: People who are immunocompromised should consult a doctor before using Xerese, as the benefit in this population has not been adequately proven.
  • Older adults (65+): There were too few patients over 65 in clinical studies to draw firm conclusions, though available results were similar to those of younger patients.
  • Skin conditions that mimic cold sores: If you are unsure whether your lesion is a cold sore, check with your doctor before using Xerese.
🚑If you take too much

An overdose from applying Xerese to the skin is unlikely, because the amount absorbed into the bloodstream through topical use is minimal. If you or someone else accidentally swallows Xerese, contact Poison Control or seek medical attention right away.

🔬Pharmacokinetics — how your body processes it

After applying Xerese to the skin, blood levels of acyclovir and hydrocortisone were not measured in studies, so the exact amount absorbed is not known. In general, topical corticosteroids like hydrocortisone can be absorbed through intact skin, and that absorption increases when the skin is broken or inflamed — both of which can occur with cold sores. Once absorbed, hydrocortisone is processed similarly to other corticosteroids: it is broken down mainly in the liver and cleared by the kidneys, with some elimination through bile as well. Overall systemic exposure from topical use on a small area is expected to be low.

📦How to store it

Store at controlled room temperature 20° to 25°C (68° to 77°F); excursions permitted to 15° to 30°C (59° to 86°F). Do not freeze.

📄 Written from Acyclovir / Hydrocortisone’s FDA-approved label information, summarized in plain language with AI, and reviewed by our pharmacy team before publication. Every point is grounded in that labeling — nothing is invented. How we use AI →

🩺 Pharmacist Counseling Corner

Quick, plain-English answers to the questions patients ask most about Acyclovir / Hydrocortisone — the kind of thing our pharmacy team would talk through with you at the counter.

What exactly does Xerese do for a cold sore?
Xerese works on two fronts. The acyclovir in it is an antiviral that stops the herpes virus from multiplying, which helps limit how bad the sore gets. The hydrocortisone is a mild anti-inflammatory that helps reduce the redness and swelling. Together, they're designed to lower the chance that your cold sore turns into an open ulcer and to help it heal faster — but starting it early (at the first tingle or redness) makes a real difference.
When is the best time to start using it?
As soon as possible — ideally the moment you feel that familiar tingling or itching, even before a visible sore appears. That early window is when antiviral treatment does the most good. Waiting until the sore is already fully developed will make it less effective.
How do I apply it correctly?
Apply a thin layer of Xerese to the sore and a little bit of the surrounding skin five times a day for five days. Try not to rub the area more than you need to — rubbing can irritate the skin and may spread the virus to other areas. It's for the lips and skin around the mouth only; keep it away from your eyes, inside your mouth, your nose, and your genitals.
Can I use Xerese if I'm pregnant or breastfeeding?
There isn't a lot of data specific to Xerese in pregnancy or breastfeeding, but because it's applied to a small area of skin, the amount that gets absorbed into your body is expected to be very low. Published data on similar topical products haven't shown a link to birth defects or pregnancy problems. That said, always tell your doctor you're pregnant or nursing so they can weigh the benefits and any risks for your specific situation.
What side effects should I watch for — and when should I call my doctor?
The most common issues are minor skin irritation, dryness, or an allergic-type reaction right where you're applying the cream. Those are usually manageable. Call your doctor if the sore hasn't started healing after two weeks — some skin infections can look just like a cold sore and need different treatment. Also reach out if you notice a severe skin reaction or worsening symptoms that don't improve.
Is it safe to use if I have a weakened immune system?
That's something to discuss with your doctor before starting Xerese. Studies in people with HIV and stable immune function showed healing times were similar to another acyclovir product, but the data weren't strong enough to confirm a clear benefit in immunocompromised patients overall. Your doctor can help figure out the best approach for treating your cold sores safely.
Is Acyclovir / Hydrocortisone available over the counter?
Acyclovir / Hydrocortisone is dispensed by prescription according to its FDA labeling, so it isn't sold over the counter. Your prescriber and pharmacist will determine if it's appropriate for you.
When was Acyclovir / Hydrocortisone first available?
Acyclovir / Hydrocortisone has been available in the United States since at least 2009, based on FDA approval history (Drugs@FDA) and product marketing records.

💬 Answers drafted from Acyclovir / Hydrocortisone’s FDA-approved label information, summarized in plain language with AI, and reviewed by our pharmacy team before publication. Grounded in that labeling — nothing is made up. How we use AI →

🧰 Keep exploring

💊 How Acyclovir / Hydrocortisone comes

Acyclovir / Hydrocortisone is available in 1 form. Different forms and brands can have different approved uses, doses, schedules, and directions. Follow the instructions for your exact product, and do not switch forms without guidance from your prescriber or pharmacist.

Topical cream, ointment or gel

On the skin
Brands Xerese
How this form is used
What it may be used for
  • Xerese is used for the early treatment of recurrent herpes labialis (cold sores) on the lips and around the mouth in adults and children 6 years and older.
  • Xerese reduces the likelihood that a cold sore will develop into an open ulcer.
  • Xerese helps shorten the time it takes for a cold sore to heal.
Important instructions
  • Xerese is applied to the skin five times a day for five days.
  • Start Xerese as early as possible — at the first sign of tingling, redness, or a lesion.
  • Apply enough Xerese to cover the sore and its outer margin; avoid unnecessary rubbing.
  • Xerese is for external use on lips and surrounding skin only — do not use in the eye, inside the mouth or nose, or on the genitals.
Available strengths 1 strength
1 FDA-listed product record

📊 Acyclovir / Hydrocortisone across the U.S. market

How Acyclovir / Hydrocortisone appears in the FDA’s National Drug Code Directory — including its dosage forms, strengths, brand names, manufacturers, and FDA-listed product records. These are directory records, not sales or prescription volume.

1
Dose forms
1
Manufacturers
1
Brand names
1
FDA-listed product records
2009
First marketed

📈 How widely Acyclovir / Hydrocortisone is used

A general measure of how commonly Acyclovir / Hydrocortisone is prescribed, based on Medicaid — one of the largest public drug programs. The figure below is prescriptions filled in Q1–Q4 2025, summed across every form and brand of the drug.

Think of this as a proxy for how widely Acyclovir / Hydrocortisone is used, drawn from freely available public data. Medicaid is just one program — these numbers don’t include Medicare, other government coverage, or commercial and cash-pay prescriptions, so real-world use is higher than what’s shown here.

11
Medicaid prescriptions filled (Q1–Q4 2025)
$13,119 gross Medicaid reimbursement (before mandatory rebates — net cost is lower)

How commonly is Acyclovir / Hydrocortisone prescribed? Of the 1,596 medications we measure, Acyclovir / Hydrocortisone ranks #1,592 by Medicaid prescriptions — more than 0% of them.

Where Acyclovir / Hydrocortisone ranks among the drugs we measure · Q1–Q4 2025 · neighbors ±5

Utilization by Acyclovir / Hydrocortisone product

Pick a product to see its own Medicaid numbers. Each chip is one clinical product — a specific strength & dosage form as defined by RxNorm — with brand-name and generic versions combined.

acyclovir 50 MG/ML / hydrocortisone 10 MG/ML Topical Cream

11 Medicaid prescriptions (Q1–Q4 2025) 100% of Acyclovir / Hydrocortisone prescriptions shown $13,119 gross reimbursement (before rebates) ≈ $1,193 per prescription (gross)

Summed across the 1 of 2 listed NDC products with Medicaid activity — every brand and generic of this exact strength & form. RxNorm 998422

Shares are of the Medicaid prescriptions shown here. Product grouping follows RxNorm (the National Library of Medicine’s drug terminology), so “one product” means one strength & dosage form regardless of manufacturer. Dollar figures are gross Medicaid reimbursement before mandatory rebates — rebates (often large, especially for brand-name drugs) are confidential, so actual net cost to Medicaid is lower than shown.

Source: Medicaid State Drug Utilization Data (CMS), aggregated by generic ingredient — summed across every NDC (all brands, strengths, salt forms and dosage forms) of Acyclovir / Hydrocortisone, and across all states and both fee-for-service and managed-care claims. A general popularity signal; it excludes Medicare, commercial insurance and cash prescriptions, so it is not total U.S. use. Based on the 1 of 2 listed Acyclovir / Hydrocortisone NDCs with Medicaid activity.

🔍 Compare Acyclovir / Hydrocortisone products

A representative set of FDA-listed product records for Acyclovir / Hydrocortisone — across manufacturers, strengths, and dosage forms, grouped by form with each product’s manufacturer and how the FDA approved it. The same medicine may be made and packaged by different companies, so a single drug can have many directory entries. (It’s also why a refill can look different — a new shape, color, or box — even though it contains the same medication.)

Strength Route Manufacturer / Labeler Category Details
💊Topical cream, ointment or gel
ACYCLOVIR 50 mg/g; HYDROCORTISONE 10 mg/g Topical Bausch Health US LLC NDA View NDC →

Showing 1 of 1 products — FDA National Drug Code Directory. See every product, package size and price: browse all 1 Acyclovir / Hydrocortisone NDCs →

RxNorm Concept Web — From Ingredient to Every Form and Strength

This page starts with one exact multiple-ingredient concept (MIN). The branches below show its dose-form concepts (SCDF), then the available clinical drug and strength concepts (SCD). A product with a different ingredient combination belongs on a different page.

Multiple ingredients (MIN) Acyclovir / Hydrocortisone RxCUI 1007804 1 dose form · 1 strength

Look up RxCUI 1007804 in the RxCUI Atlas →

RxNorm is the U.S. National Library of Medicine’s normalized drug vocabulary. Its concept hierarchy can include forms that are not currently marketed; the status on each branch compares that concept with current FDA listings. RxCUIs identify vocabulary concepts, not individual packages or manufacturers.

🏷️ Sold under these brand names

Xerese

🏭 Manufacturers & labelers

Bausch Health US LLC 1

RxNorm drug class

Acyclovir / Hydrocortisone belongs to the Herpesvirus Nucleoside Analog DNA Polymerase Inhibitor class.

Pharmacologic class Herpesvirus Nucleoside Analog DNA Polymerase Inhibitor, Herpes Simplex Virus Nucleoside Analog DNA Polymerase Inhibitor, Herpes Zoster Virus Nucleoside Analog DNA Polymerase Inhibitor
Drug family (ATC) Antivirals, Nucleosides and nucleotides excl. reverse transcriptase inhibitors, Antivirals
How it works DNA Polymerase Inhibitors

Classified by RxNorm RxClass — the U.S. National Library of Medicine's standardized drug-classification service (Established Pharmacologic Class from the FDA, the ATC drug family from the WHO, and mechanism of action). Reference only, not medical advice.

🔬 Where this comes from

Core label, product, RxNorm, safety, and utilization data on this page come from the sources identified below. AI-written, editorial, and licensed sections are labeled separately.

📄
FDA-filed drug labels (SPL) Uses, dosing, warnings & side effects from SPL records retrieved through openFDA; the linked representative set can be verified on DailyMed. ✓ Linked label effective Aug 3, 2020
🏭
Forms, brands & labelersAggregated from ingredient-matched FDA National Drug Code Directory product records for Acyclovir / Hydrocortisone.
📈
Real-world reportsThe FDA Adverse Event Reporting System (FAERS), served through openFDA.
🚨
Recalls & shortagesopenFDA drug-enforcement reports and the FDA drug-shortage database.
🧾 Clinical label set — FDA-filed SPL labels retained for Acyclovir / Hydrocortisone after exact ingredient or ingredient-combination matching and applicable route/form matching
Clinical labels in scope
1
NDC products indexed
1
Distinct labelers/manufacturers represented
1
Linked representative label
Bausch Health US LLC
Linked label effective
Aug 3, 2020
Composite sections available
20
Linked SPL Set ID
3b6ac164-0f1e-4f36-94a1-1fdb07d710f5
Linked SPL Document ID
a4efb63c-e7bf-43da-bbfe-463f672cb1bc
Open the linked representative label on DailyMed ↗
NDC package records associated with this linked SPL 1

How we combine label and product data

HelloPharmacist combines public FDA and NLM records; we don’t author the underlying clinical facts. We identified 1 FDA-filed SPL label set within the page’s selected clinical scope after exact ingredient or ingredient-combination matching and applicable route/form matching. The representative label is the starting point for the displayed reference monograph; the 12 largest stored in-scope SPL records, which may include that representative, are compared section by section, and the longest available version of each section is retained. Forms, routes, brands, labelers, product-listed strengths, and product-record counts are aggregated separately from ingredient-matched FDA NDC Directory records; package records listed above are associated with the linked SPL; and the normalized concept hierarchy comes from NLM RxNorm.

For canonical ingredient pages, bounded product-attributed indication and administration excerpts may be added to the AI evidence, and the generator is instructed to preserve available product, brand, route, and form qualifiers instead of treating one label as universal. Where a section is identified as AI-written, its plain-language text is generated from bounded label evidence. New draft drug pages remain in the admin review queue before first publication. Bausch Health US LLC is the representative DailyMed label linked for verification and dates; it is not the sole source used for the page.

This is general education, not medical advice — always consult your doctor or pharmacist about your medications and any medical condition. For the exact wording of the linked representative label, view that label on DailyMed; some displayed composite sections may come from other in-scope SPL labels. Learn how we use AI and our data sources & update cadence.