Avacopan

107 interactions 11 explained in plain English
Also sold as: Tavneos
Dr. Brian Staiger, PharmD, BCPS
Medically reviewed by Dr. Brian Staiger, PharmD, BCPS · Updated Jul 4, 2026 · Editorial policy · Data sources

Sources: FDA prescribing information (Structured Product Labeling), the published literature cited in each entry, DDInter 2.0 (a major open-access drug-interaction database), and legacy DrugBank interaction data distributed by the NIH's RxNav service (decommissioned in 2024) — analyzed and reviewed by our pharmacist team. How we build this library →

Major

Avacopan Acetaminophen And Codeine Capital® & Codeine Explained Increased codeine and morphine exposure Details Avacopan Clindamycin ANTIROBE Explained Increased exposure to CYP3A4 substrate Details Avacopan Omeprazole Gastrobim Explained Increased CYP3A4 substrate exposure Details Avacopan Sertraline Explained Increased CYP3A4 substrate exposure Details Avacopan Buprenorphine Belbuca Explained Increased CYP3A4 substrate exposure Details Avacopan Colchicine Colcrys Explained Increased exposure to CYP3A4 substrate Details Avacopan Simvastatin Flolipid Explained Increased simvastatin exposure Details Avacopan Abemaciclib Verzenio Explained Increased exposure to CYP3A4 substrate Details Avacopan Acalabrutinib Calquence Increased exposure to CYP3A4 substrate Details Avacopan Apixaban Eliquis Explained Increased CYP3A4 substrate exposure Details Avacopan Aripiprazole Injection Abilify Increased CYP3A4 substrate exposure Details Avacopan Asciminib Scemblix Increased CYP3A4 substrate exposure Details Avacopan Avapritinib Ayvakit Increased CYP3A4 substrate exposure Details Avacopan Avatrombopag Doptelet Increased CYP3A4 substrate exposure Details Avacopan Belumosudil Rezurock Explained Increased CYP3A4 substrate exposure Details Avacopan Atorvastatin Atorvaliq Increased CYP3A4 substrate exposure Details Avacopan Cariprazine Vraylar Explained Increased CYP3A4 substrate exposure Details Avacopan Abiraterone Abirtega Increased CYP3A4 substrate exposure Details Avacopan Alfuzosin UroXatral Increased CYP3A4 substrate exposure Details Avacopan Amlodipine Amvaz® Increased CYP3A4 substrate exposure Details Avacopan Avanafil Stendra Increased CYP3A4 substrate exposure Details Avacopan Axitinib Inlyta Increased exposure to CYP3A4 substrate Details Avacopan Bedaquiline Sirturo Increased CYP3A4 substrate exposure Details Avacopan Bosutinib Bosulif Increased exposure to CYP3A4 substrate Details Avacopan Brexpiprazole Rexulti Increased CYP3A4 substrate exposure Details Avacopan Brigatinib Alunbrig Increased exposure to CYP3A4 substrate Details Avacopan Budesonide Entocort Increased budesonide exposure Details Avacopan Budesonide Nasal Spray Rhinocort Increased budesonide exposure Details Avacopan Budesonide Oral Inhalation Pulmicort Increased budesonide exposure Details Avacopan Cabozantinib Cabometyx Increased CYP3A4 substrate exposure Details Avacopan Cabozantinib (Thyroid Cancer) Cabometyx Increased CYP3A4 substrate exposure Details Avacopan Capmatinib Tabrecta Increased CYP3A4 substrate exposure Details Avacopan Clindamycin Injection ANTIROBE Increased exposure to CYP3A4 substrate Details Avacopan Clindamycin Topical C/T/S® Increased exposure to CYP3A4 substrate Details Avacopan Clindamycin Vaginal Cleocin Increased exposure to CYP3A4 substrate Details Avacopan Cobimetinib Cotellic Increased exposure to CYP3A4 substrate Details Avacopan Cyclosporine Injection Atopica Increased exposure to CYP3A4 substrate Details Avacopan Cyclosporine Ophthalmic Cequa Increased exposure to CYP3A4 substrate Details Avacopan Darolutamide Nubeqa Increased CYP3A4 substrate exposure Details Avacopan Dasatinib Phyrago Increased exposure to CYP3A4 substrate Details

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