Cilostazol

78 interactions 8 explained in plain English
Also sold as: Pletal®
About Cilostazol

Cilostazol is an antiplatelet medication used to reduce leg pain caused by poor blood flow during walking. Read the full Cilostazol drug information page →

Dr. Brian Staiger, PharmD, BCPS
Medically reviewed by Dr. Brian Staiger, PharmD, BCPS · Updated Jun 30, 2026 · Editorial policy · Data sources

Sources: FDA prescribing information (Structured Product Labeling), the published literature cited in each entry, DDInter 2.0 (a major open-access drug-interaction database), and legacy DrugBank interaction data distributed by the NIH's RxNav service (decommissioned in 2024) — analyzed and reviewed by our pharmacist team. How we build this library →

Major

Cilostazol Acetaminophen And Codeine Capital® & Codeine Explained Increased codeine and morphine exposure Details Cilostazol Abametapir Explained Increased exposure of CYP3A4 substrate Details Cilostazol Omeprazole Gastrobim Explained Increased cilostazol exposure Details Cilostazol Sertraline Explained An increased risk of bleeding Details Cilostazol Colchicine Colcrys Explained Increased colchicine exposure and an increased risk of colchicine-related toxicity Details Cilostazol Apixaban Eliquis Explained Increased risk of bleeding and can cause serious, potentially fatal bleeding Details Cilostazol Aspirin Acuprin® An increased risk of bleeding Details Cilostazol Aspirin Rectal Aspirin An increased risk of bleeding Details Cilostazol Betrixaban Bevyxxa® Increased risk of bleeding Details Cilostazol Abiraterone Abirtega Increased cilostazol exposure Details Cilostazol Anagrelide Agrylin Increased bleeding risk; additive vasodilation; increased risk of tachycardia, palpitations, and heart failure Details Cilostazol Bedaquiline Sirturo Increased bedaquiline exposure Details Cilostazol Bromfenac Ophthalmic Bromday® An increased risk of bleeding Details Cilostazol Budesonide Entocort Increased budesonide exposure Details Cilostazol Budesonide Nasal Spray Rhinocort Increased budesonide exposure Details Cilostazol Budesonide Oral Inhalation Pulmicort Increased budesonide exposure Details Cilostazol Caplacizumab-Yhdp Injection Cablivi An increased risk of bleeding Details Cilostazol Clopidogrel Plavix An increased risk of bleeding Details Cilostazol Dabigatran Pradaxa® Increased risk of bleeding Details Cilostazol Dabigatran Etexilate Increased risk of bleeding Details Cilostazol Diclofenac Ophthalmic Voltaren® Eye Drops An increased risk of bleeding Details Cilostazol Diclofenac Topical (Actinic Keratosis) Pennsaid An increased risk of bleeding Details Cilostazol Diclofenac Topical (Arthritis Pain) Pennsaid® An increased risk of bleeding Details Cilostazol Diclofenac Transdermal Patch Flector An increased risk of bleeding Details Cilostazol Dipyridamole Permole® An increased risk of bleeding Details Cilostazol Doxorubicin Adriamycin Increased doxorubicin exposure and an increased risk of doxorubicin-related adverse reactions Details Cilostazol Edoxaban Savaysa Increased risk of bleeding Details Cilostazol Esomeprazole Nexium Increased cilostazol exposure Details Cilostazol Esomeprazole Injection Nexium Increased cilostazol exposure Details Cilostazol Etodolac Lodine An increased risk of bleeding Details Cilostazol Fenoprofen Fenopron An increased risk of bleeding Details Cilostazol Fentanyl Transdermal Patch Duragesic® Increased fentaNYL exposure and an increased risk of prolonged opioid effects Details Cilostazol Finerenone Kerendia Increased finerenone exposure and an increased risk of finerenone-related adverse effects Details Cilostazol Flurbiprofen Ansaid An increased risk of bleeding Details Cilostazol Flurbiprofen Ophthalmic Ocufen An increased risk of bleeding Details Cilostazol Fondaparinux Arixtra Increased risk of bleeding Details Cilostazol Fondaparinux Injection Arixtra Increased risk of bleeding Details Cilostazol Heparin Increased risk of bleeding Details

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Educational information only, not medical advice. Always confirm interactions with your pharmacist or prescriber before making any change to your medications.