FDA-filed SPL labeling · retrieved through openFDA

Heparin / Taurolidine

Heparin/taurolidine is an antimicrobial and anticoagulant combination used to reduce catheter-related bloodstream infections in adults with kidney failure on chronic hemodialysis.

Brand name Defencath
Drug classes Anti-coagulant
Rx Form 1 Route Intraluminal
Dr. Brian Staiger, PharmD, BCPS
Reviewed by Last reviewed Aug 28, 2026
🧬 Where this information comes from Click to expand

The clinical label records used on this page are FDA-filed Structured Product Labeling (SPL) retrieved through openFDA. We identified 1 clinical label set within the page’s selected clinical scope after exact ingredient or ingredient-combination matching and applicable route/form matching. Forms, routes, brands, labelers, strengths, and NDC product-record counts are built separately from matching FDA National Drug Code Directory records. The linked DailyMed document is a representative official source for verification, not the page’s only clinical source. View the linked label on DailyMed →

At a glance
Linked label effectiveSep 4, 2026
AvailabilityRx
Earliest approval/marketing year 2024
FDA-listed product records 6
Boxed warningNone found in compared labels
How we combine label and product data →
No current FDA shortage listed · checked Sep 20, 2026
Heparin / Taurolidine at a glance The quick version — the full detail is in the Patient Information Guide below.
💊
HelloPharmacist Editorial Team Bottom Line
Defencath is a catheter lock solution — not an injection or oral medication — used to protect the central venous catheter of adult kidney failure patients on chronic hemodialysis from serious bloodstream infections. It is instilled into the catheter after each dialysis session and removed before the next one. The most important risks to watch for are signs of a heparin-related platelet reaction (HIT) or an allergic reaction, both of which require stopping the medication immediately.

📖 Heparin / Taurolidine: Patient Information Guide

A plain-language walkthrough of Heparin / Taurolidine — what it treats, how it works, how it’s taken, side effects, warnings and interactions. Tap any section to expand it.

🎯What it's used for

Heparin/taurolidine is an antimicrobial and anticoagulant combination used as a catheter lock solution in a specific patient population.

  • Defencath (intraluminal route) is approved to reduce the risk of catheter-related bloodstream infections (CRBSIs) in adults with kidney failure receiving chronic hemodialysis through a central venous catheter (CVC)
  • Defencath is approved for use in this limited and specific population only — its safety and effectiveness have not been established for other patients or other uses
⚙️How it works

Defencath works through two different mechanisms. Taurolidine, the antimicrobial component, damages bacterial cell walls and prevents bacteria from sticking to the inside surfaces of the catheter. Heparin, the anticoagulant component, activates a blood protein called Antithrombin III, which then blocks key clotting factors (especially Factor Xa and thrombin/Factor IIa) from forming clots. Heparin also prevents a stable fibrin clot from forming by blocking the fibrin-stabilizing factor — though it cannot dissolve clots that have already formed.

Because Defencath sits inside the catheter rather than circulating through the body, it acts locally to protect the catheter between dialysis sessions.

💊How it's taken

Defencath is not taken by mouth or given as an injection into a vein. It is instilled directly into the lumens (internal channels) of a central venous catheter by a healthcare provider at the end of each hemodialysis session.

  • The solution remains inside the catheter between sessions and is aspirated (drawn out) and discarded before the next session begins
  • Each single-dose vial is intended for one patient and one use — any leftover solution must be discarded
  • If the solution cannot be aspirated before the next session, standard catheter care should be followed and the catheter checked for problems
🤒Side effects — in detail

The most frequently reported side effects in clinical trials of Defencath (occurring in 2% or more of patients) included:

  • Hemodialysis catheter malfunction
  • Hemorrhage or bleeding (including at various sites such as the gastrointestinal tract, catheter site, and urinary tract)
  • Nausea
  • Vomiting
  • Dizziness
  • Musculoskeletal chest pain (non-cardiac chest discomfort)
  • Low platelet count (thrombocytopenia)
  • Low calcium levels (hypocalcemia) — less than 1% of patients
  • Altered taste (dysgeusia) — less than 1% of patients
  • Numbness or tingling (paresthesia) — reported in post-marketing use outside the US

Serious reactions to watch for and report immediately include signs of heparin-induced thrombocytopenia (HIT) — such as unusual bruising or unexpected clotting — and signs of an allergic reaction such as rash, swelling, or breathing difficulty.

⚠️Warnings & precautions
  • Heparin-Induced Thrombocytopenia (HIT): A rare but serious immune reaction to heparin that causes a dangerous drop in platelets and can lead to blood clots. HIT occurred in about 0.3% of patients in clinical trials. If HIT develops, Defencath must be stopped right away and treated promptly. Defencath is contraindicated in anyone with a known history of HIT.
  • Drug Hypersensitivity (Allergic Reactions): Allergic reactions to heparin or other components of Defencath were reported in about 0.5% of clinical trial patients. If any allergic reaction occurs, Defencath should be stopped and medical care sought immediately. Defencath is contraindicated in patients with known hypersensitivity to taurolidine, heparin, citrate, or pork products.
🔀What it interacts with

The FDA label for Defencath does not identify specific drug, food, or supplement interactions.

This is not a complete list of interactions. Always talk with your doctor or pharmacist before starting, stopping, or changing any medication.

📋Before taking it
  • Do not use Defencath if you have ever had heparin-induced thrombocytopenia (HIT)
  • Do not use Defencath if you are allergic to taurolidine, heparin, citrate, or pork products
  • Defencath has not been approved for use in children — safety and effectiveness in pediatric patients have not been established
  • Pregnant patients: Defencath is not intended to enter the bloodstream, so fetal exposure is not expected, but inform your care team if you are pregnant
  • Breastfeeding patients: Because Defencath stays inside the catheter and is not absorbed systemically, infant exposure through breast milk is not expected — still, inform your care team
  • Older adults (65 and over): Clinical trial data showed no meaningful difference in safety or effectiveness compared to younger adults
📡Pharmacodynamics — effects in the body

The overall pharmacodynamic effects of Defencath in the body are not fully characterized. The taurolidine component has been shown in laboratory studies to kill bacteria (bactericidal activity) by damaging microbial cell walls and preventing bacteria from adhering to biological surfaces. Heparin within the catheter blocks key steps in the blood-clotting process, helping to prevent clot formation inside the catheter lumen.

🔬Pharmacokinetics — how your body processes it

No pharmacokinetic studies (studies measuring how the drug is absorbed, distributed, metabolized, and eliminated) were conducted for Defencath. Because it is designed to be instilled only into the catheter lumens and is not intended for systemic administration, it is not expected to circulate through the body in meaningful amounts.

📦How to store it

stored at a controlled room temperature of 20°C to 25°C (68°F to 77°F); excursions are permitted from 15°C to 30°C (59°F to 86°F) . Do not freeze. stored in the commercial carton, prior to the instillation in central venous catheters.

📄 Written from Heparin / Taurolidine’s FDA-approved label information, summarized in plain language with AI, and reviewed by our pharmacy team before publication. Every point is grounded in that labeling — nothing is invented. How we use AI →

🩺 Pharmacist Counseling Corner

Quick, plain-English answers to the questions patients ask most about Heparin / Taurolidine — the kind of thing our pharmacy team would talk through with you at the counter.

What exactly is Defencath and why has my doctor prescribed it?
Defencath is a special solution placed inside your dialysis catheter after each hemodialysis session to help prevent serious infections in the bloodstream. When you're on long-term dialysis through a central venous catheter, that catheter can become a pathway for bacteria to enter your bloodstream — Defencath works to stop that. It contains two ingredients: taurolidine (which kills bacteria inside the catheter) and heparin (which prevents clots from forming in the catheter between sessions).
How is Defencath given — do I take a pill or get an injection?
Neither, actually. Defencath is instilled directly into the channels of your dialysis catheter by your healthcare team at the end of each dialysis session. It stays inside the catheter while you're home between sessions. Before your next session begins, the care team draws it out and discards it — it doesn't get flushed into your body. You don't swallow it, and it's not injected into your veins.
What side effects should I watch out for and when should I call someone?
The most common issues reported in clinical trials included catheter malfunction, some bleeding or bruising, nausea, vomiting, dizziness, and chest muscle discomfort. Most of these are manageable, but two reactions need prompt attention: if you notice unusual bruising, a sudden drop in platelet count, or unexpected blood clots forming, that could be a sign of a rare reaction called heparin-induced thrombocytopenia (HIT) — call your care team right away. Also, any signs of an allergic reaction (rash, swelling, trouble breathing) mean you should get medical help immediately.
Is Defencath safe if I'm pregnant or breastfeeding?
Since Defencath is locked inside the catheter and not designed to travel through your bloodstream, it's not expected to reach a developing baby or pass into breast milk. That said, always let your care team know if you are pregnant or breastfeeding so they can make the best decision for your situation.
I've had a bad reaction to heparin before — can I still use Defencath?
This is really important to tell your doctor before starting Defencath. If you've ever been diagnosed with heparin-induced thrombocytopenia (HIT) — the serious immune reaction to heparin — Defencath is contraindicated, meaning it should not be used at all. The same applies if you're allergic to taurolidine, heparin, citrate, or pork products. Your care team will need to find an alternative approach for protecting your catheter.
What happens if the solution can't be removed from my catheter before my next dialysis session?
Your care team is trained for this situation. If Defencath can't be aspirated (drawn out) before the next session, they'll follow standard catheter care procedures and flush the catheter with normal saline. If there's a sign of catheter malfunction, they'll take the appropriate next steps. It's important not to try to flush the solution in yourself — always leave catheter management to your healthcare team.
Is Heparin / Taurolidine available over the counter?
Heparin / Taurolidine is dispensed by prescription according to its FDA labeling, so it isn't sold over the counter. Your prescriber and pharmacist will determine if it's appropriate for you.
When was Heparin / Taurolidine first available?
Heparin / Taurolidine has been available in the United States since at least 2024, based on FDA approval history (Drugs@FDA) and product marketing records.
Who makes Heparin / Taurolidine?
Heparin / Taurolidine is supplied by 2 manufacturers listed in the FDA NDC Directory, including CorMedix Inc., ROVI Pharma Industrial Services SA.

💬 Answers drafted from Heparin / Taurolidine’s FDA-approved label information, summarized in plain language with AI, and reviewed by our pharmacy team before publication. Grounded in that labeling — nothing is made up. How we use AI →

🧰 Keep exploring

💊 How Heparin / Taurolidine comes

Heparin / Taurolidine is available in 1 form. Different forms and brands can have different approved uses, doses, schedules, and directions. Follow the instructions for your exact product, and do not switch forms without guidance from your prescriber or pharmacist.

Oral solution

By mouth · Intraluminal
Brands Defencath
How this form is used
What it may be used for
  • Defencath is used to reduce the incidence of catheter-related bloodstream infections (CRBSIs) in adults with kidney failure receiving chronic hemodialysis through a central venous catheter
Important instructions
  • Defencath is instilled into each lumen of the central venous catheter at the conclusion of each hemodialysis session — it is not given by mouth or injected into a vein
  • Defencath should be aspirated from the catheter and discarded before the next hemodialysis session begins
  • Defencath must not be used as a catheter flush product and is not intended for systemic (whole-body) administration
  • Each Defencath single-dose vial is for one patient and one instillation only — discard any unused portion remaining in the vial
Available strengths 5 strengths
6 FDA-listed product records

📊 Heparin / Taurolidine across the U.S. market

How Heparin / Taurolidine appears in the FDA’s National Drug Code Directory — including its dosage forms, strengths, brand names, manufacturers, and FDA-listed product records. These are directory records, not sales or prescription volume.

1
Dose forms
2
Manufacturers
1
Brand names
6
FDA-listed product records
2024
First marketed
CorMedix Inc.67%
ROVI Pharma Industrial Services SA33%

Share of FDA-listed product records by manufacturer — FDA National Drug Code Directory. Record counts are not sales or prescription volume.

📈 How widely Heparin / Taurolidine is used

A general measure of how commonly Heparin / Taurolidine is prescribed, based on Medicaid — one of the largest public drug programs. The figure below is prescriptions filled in Q1–Q4 2025, summed across every form and brand of the drug.

Think of this as a proxy for how widely Heparin / Taurolidine is used, drawn from freely available public data. Medicaid is just one program — these numbers don’t include Medicare, other government coverage, or commercial and cash-pay prescriptions, so real-world use is higher than what’s shown here.

1,550
Medicaid prescriptions filled (Q1–Q4 2025)
$194,461 gross Medicaid reimbursement (before mandatory rebates — net cost is lower)

How commonly is Heparin / Taurolidine prescribed? Of the 1,596 medications we measure, Heparin / Taurolidine ranks #1,221 by Medicaid prescriptions — more than 23% of them.

Where Heparin / Taurolidine ranks among the drugs we measure · Q1–Q4 2025 · neighbors ±5

Utilization by Heparin / Taurolidine product

Pick a product to see its own Medicaid numbers. Each chip is one clinical product — a specific strength & dosage form as defined by RxNorm — with brand-name and generic versions combined.

3 ML heparin sodium, porcine 1000 UNT/ML / taurolidine 13.5 MG/ML Injection

1,550 Medicaid prescriptions (Q1–Q4 2025) 100% of Heparin / Taurolidine prescriptions shown $194,461 gross reimbursement (before rebates) ≈ $125 per prescription (gross)

Summed across the 1 of 2 listed NDC products with Medicaid activity — every brand and generic of this exact strength & form. RxNorm 2670461

Shares are of the Medicaid prescriptions shown here. Product grouping follows RxNorm (the National Library of Medicine’s drug terminology), so “one product” means one strength & dosage form regardless of manufacturer. Dollar figures are gross Medicaid reimbursement before mandatory rebates — rebates (often large, especially for brand-name drugs) are confidential, so actual net cost to Medicaid is lower than shown.

Source: Medicaid State Drug Utilization Data (CMS), aggregated by generic ingredient — summed across every NDC (all brands, strengths, salt forms and dosage forms) of Heparin / Taurolidine, and across all states and both fee-for-service and managed-care claims. A general popularity signal; it excludes Medicare, commercial insurance and cash prescriptions, so it is not total U.S. use. Based on the 1 of 2 listed Heparin / Taurolidine NDCs with Medicaid activity.

🔍 Compare Heparin / Taurolidine products

A representative set of FDA-listed product records for Heparin / Taurolidine — across manufacturers, strengths, and dosage forms, grouped by form with each product’s manufacturer and how the FDA approved it. The same medicine may be made and packaged by different companies, so a single drug can have many directory entries. (It’s also why a refill can look different — a new shape, color, or box — even though it contains the same medication.)

Strength Route Manufacturer / Labeler Category Details
💊Oral solution
TAUROLIDINE 40.5 mg/3 mL; HEPARIN 3000 [USP'U]/3 mL Intraluminal CorMedix Inc. × 2 listings NDA View NDC →
3000; 40.5 [USP'U]/3 mL; mg/3 mL Intraluminal CorMedix Inc. NDA View NDC →
5000; 67.5 [USP'U]/5 mL; mg/5 mL Intraluminal CorMedix Inc. NDA View NDC →
HEPARIN 3000 [USP'U]/3 mL; TAUROLIDINE 40.5 mg/3 mL ROVI Pharma Industrial Services SA DRUG FOR FURTHER PROCESSING View NDC →
HEPARIN 5000 [USP'U]/5 mL; TAUROLIDINE 67.5 mg/5 mL ROVI Pharma Industrial Services SA DRUG FOR FURTHER PROCESSING View NDC →

Showing 6 of 6 products — FDA National Drug Code Directory. See every product, package size and price: browse all 6 Heparin / Taurolidine NDCs →

RxNorm Concept Web — From Ingredient to Every Form and Strength

This page starts with one exact multiple-ingredient concept (MIN). The branches below show its dose-form concepts (SCDF), then the available clinical drug and strength concepts (SCD). A product with a different ingredient combination belongs on a different page.

Multiple ingredients (MIN) Heparin / Taurolidine RxCUI 2670456 1 dose form · 1 strength

Look up RxCUI 2670456 in the RxCUI Atlas →

RxNorm is the U.S. National Library of Medicine’s normalized drug vocabulary. Its concept hierarchy can include forms that are not currently marketed; the status on each branch compares that concept with current FDA listings. RxCUIs identify vocabulary concepts, not individual packages or manufacturers.

🏷️ Sold under these brand names

Defencath

🏭 Manufacturers & labelers

CorMedix Inc. 4 ROVI Pharma Industrial Services SA 2

RxNorm drug class

Heparin / Taurolidine belongs to the Antiinfectives class.

Drug family (ATC) Antiinfectives

Classified by RxNorm RxClass — the U.S. National Library of Medicine's standardized drug-classification service (Established Pharmacologic Class from the FDA, the ATC drug family from the WHO, and mechanism of action). Reference only, not medical advice.

🔬 Where this comes from

Core label, product, RxNorm, safety, and utilization data on this page come from the sources identified below. AI-written, editorial, and licensed sections are labeled separately.

📄
FDA-filed drug labels (SPL) Uses, dosing, warnings & side effects from SPL records retrieved through openFDA; the linked representative set can be verified on DailyMed. ✓ Linked label effective Sep 4, 2026
🏭
Forms, brands & labelersAggregated from ingredient-matched FDA National Drug Code Directory product records for Heparin / Taurolidine.
📈
Real-world reportsThe FDA Adverse Event Reporting System (FAERS), served through openFDA.
🚨
Recalls & shortagesopenFDA drug-enforcement reports and the FDA drug-shortage database.
🧾 Clinical label set — FDA-filed SPL labels retained for Heparin / Taurolidine after exact ingredient or ingredient-combination matching and applicable route/form matching
Clinical labels in scope
1
NDC products indexed
6
Distinct labelers/manufacturers represented
2
Linked representative label
CorMedix Inc.
Linked label effective
Sep 4, 2026
Composite sections available
19
Linked SPL Set ID
13b3a61e-5a4b-4afb-8fa1-d76ebdb344d6
Linked SPL Document ID
c4c34743-4c50-4dd2-836c-3669dcdcb349
Open the linked representative label on DailyMed ↗

How we combine label and product data

HelloPharmacist combines public FDA and NLM records; we don’t author the underlying clinical facts. We identified 1 FDA-filed SPL label set within the page’s selected clinical scope after exact ingredient or ingredient-combination matching and applicable route/form matching. The representative label is the starting point for the displayed reference monograph; the 12 largest stored in-scope SPL records, which may include that representative, are compared section by section, and the longest available version of each section is retained. Forms, routes, brands, labelers, product-listed strengths, and product-record counts are aggregated separately from ingredient-matched FDA NDC Directory records; package records listed above are associated with the linked SPL; and the normalized concept hierarchy comes from NLM RxNorm.

For canonical ingredient pages, bounded product-attributed indication and administration excerpts may be added to the AI evidence, and the generator is instructed to preserve available product, brand, route, and form qualifiers instead of treating one label as universal. Where a section is identified as AI-written, its plain-language text is generated from bounded label evidence. New draft drug pages remain in the admin review queue before first publication. CorMedix Inc. is the representative DailyMed label linked for verification and dates; it is not the sole source used for the page.

This is general education, not medical advice — always consult your doctor or pharmacist about your medications and any medical condition. For the exact wording of the linked representative label, view that label on DailyMed; some displayed composite sections may come from other in-scope SPL labels. Learn how we use AI and our data sources & update cadence.