Etravirine
Generic name: Pronounced as (e'' tra vir' een)
Medical Content Reviewed By HelloPharmacist Staff
Last Revised - 11/15/2018
On this page
- Why is this medication prescribed?
- How should this medicine be used?
- Other uses for this medicine
- What special precautions should I follow?
- What special dietary instructions should I follow?
- What should I do if I forget a dose?
- What side effects can this medication cause?
- What should I know about STORAGE and DISPOSAL of this medication?
- What should I do in case of OVERDOSE?
- What OTHER INFORMATION should I know?
- Drug interactions
Why is this medication prescribed?
Etravirine is used along with other medications to treat human immunodeficiency virus (HIV) infection in adults and children 2 years of age and older who no longer benefit from taking other HIV medications. Etravirine is in a class of medications called non-nucleoside reverse transcriptase inhibitors (NNRTIs). It works by decreasing the amount of HIV in the blood. Although etravirine does not cure HIV, it may decrease your chance of developing acquired immunodeficiency syndrome (AIDS) and HIV-related illnesses such as serious infections or cancer. Taking these medications along with practicing safer sex and making other lifestyle changes may decrease the risk of transmitting (spreading) the HIV virus to other people.
How should this medicine be used?
Etravirine comes as a tablet to take by mouth. It is usually taken after a meal two times a day. Take etravirine at around the same times every day. Follow the directions on your prescription label carefully, and ask your doctor or pharmacist to explain any part you do not understand. Take etravirine exactly as directed. Do not take more or less of it or take it more often than prescribed by your doctor.
Swallow the tablets whole with liquid, such as water; do not split, chew, or crush them.
If you have trouble swallowing the tablets, they may be dissolved in water. To prepare, add the tablets to one teaspoon (5 mL) of water (only water, do not use any other type of liquid) or at least enough liquid to cover the medication, and stir until a milky mixture occurs. Then add one tablespoon (15 mL) of a liquid such as water or you can use a beverage such as orange juice or milk to improve the taste. Do not mix the tablets with a warm or hot liquid or a carbonated beverage such as a soda. Drink the mixture right away. Rinse the glass with water, orange juice, or milk and swallow the entire contents. Repeat process of rinsing and swallowing the rinse mixture several times to make sure that the entire dose is taken.
Etravirine helps to control HIV infection but does not cure it. Continue to take etravirine even if you feel well. Do not stop taking etravirine without talking to your doctor. If you stop taking etravirine or miss doses, your condition may become more difficult to treat. When your supply of etravirine starts to run low, get more from your doctor or pharmacist.
Ask your pharmacist or doctor for a copy of the manufacturer's information for the patient.
Other uses for this medicine
This medication may be prescribed for other uses; ask your doctor or pharmacist for more information.
What special precautions should I follow?
Before taking etravirine,
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tell your doctor and pharmacist if you are allergic to etravirine, any other medications, or any of the ingredients in etravirine tablets. Ask your pharmacist or check the Medication Guide for a list of the ingredients.
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tell your doctor and pharmacist what other prescription and nonprescription medications, vitamins, and nutritional supplements you are taking or plan to take. Be sure to mention the following: anticoagulants ('blood thinners') such as warfarin (Coumadin, Jantoven); antiarrhythmics (medications to treat abnormal heartbeats) including amiodarone (Nexterone, Pacerone), bepridil (Vascor), disopyramide (Norpace), flecainide (Tambocor), lidocaine (Xylocaine), mexiletine (Mexitil), propafenone (Rythmol), and quinidine (Quinidex); certain medications to treat seizures such as carbamazepine (Carbatrol, Tegretol, Teril), phenobarbital (Luminal), and phenytoin (Dilantin, Phenytek); clarithromycin (Biaxin, in Prevpac); cholesterol-lowering medications (statins) including atorvastatin (Lipitor), fluvastatin (Lescol), lovastatin (Advicor, Altoprev, Mevacor), rosuvastatin (Crestor), and simvastatin (Vytorin, Zocor); clopidogrel (Plavix); diazepam (Valium); dexamethasone; certain medications that suppress the immune system such as cyclosporine (Gengraf, Neoral, Sandimmune), sirolimus (Rapamune), and tacrolimus (Prograf); medications to treat erectile dysfunction including sildenafil (Viagra), tadalafil (Cialis), and vardenafil (Levitra); medications to treat fungal infections including fluconazole (Diflucan), itraconazole (Onmel, Sporanox), ketoconazole (Nizoral), posaconazole (Noxafil), and voriconazole (Vfend); methadone (Dolophine); other medications to treat HIV including amprenavir (Agenerase), atazanavir (Reyataz), delavirdine (Rescriptor), efavirenz (Sustiva, in Atripla), fosamprenavir (Lexiva), indinavir (Crixivan), lopinavir (in Kaletra), nelfinavir (Viracept), and nevirapine (Viramune) ritonavir (Norvir, in Kaletra), and tipranavir (Aptivus); rifabutin (Mycobutin); rifampin (Rifadin, Rifater, Rifamate); and rifapentine (Priftin). Many other medications may also interact with etravirine, so be sure to tell your doctor about all the medications you are taking, even those that do not appear on this list. Do not start taking any new medications while you are taking etravirine without first talking with your doctor or pharmacist.
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tell your doctor what herbal products you are taking, especially St. John's wort.
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tell your doctor if you have or have ever had liver disease, including hepatitis.
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tell your doctor if you are pregnant or plan to become pregnant. If you become pregnant while taking etravirine, call your doctor.
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you should not breastfeed if you are infected with HIV or are taking etravirine.
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you should know that your body fat may increase or move to different areas of your body such as your breasts, neck, chest, stomach, and upper back. Loss of fat from your legs, arms, and face may also happen.
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you should know that while you are taking medications to treat HIV infection, your immune system may get stronger and begin to fight other infections that were already in your body. This may cause you to develop symptoms of those infections. If you have new or worsening symptoms after starting treatment with etravirine, be sure to tell your doctor.
What special dietary instructions should I follow?
Talk to your doctor about eating grapefruit and drinking grapefruit juice while taking this medicine.
What should I do if I forget a dose?
If you remember that you have missed taking a dose within 6 hours of the time you usually take etravirine, take the missed dose following a meal as soon as possible, and take the next dose at the regularly scheduled time. However, if you remember more than 6 hours after the time you usually take your dose, wait and take the next dose of etravirine according to your regular dosing schedule. Do not take a double dose to make up for a missed one.
What side effects can this medication cause?
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Etravirine may cause side effects. Tell your doctor if any of these symptoms are severe or do not go away:
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nausea
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vomiting
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abdominal pain
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diarrhea
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headache
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increase in blood pressure
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pain, burning, numbness, or tingling in the hands or feet
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Some side effects can be serious. If you experience any of these symptoms, stop taking etravirine and call your doctor immediately:
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rash
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redness, bumps, or blisters on the skin or in the mouth
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redness or swelling of the eyes
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swelling of the face
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sore throat, cough, fever, chills, or other signs of infection
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general ill feeling
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tiredness
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muscle or joint aches
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yellowing of the skin or eyes
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dark-colored urine
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pale-colored stools
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pain in the upper right part of the stomach
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loss of appetite
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Etravirine may cause other side effects. Call your doctor if you have any unusual problems while taking this medication.
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If you experience a serious side effect, you or your doctor may send a report to the Food and Drug Administration's (FDA) MedWatch Adverse Event Reporting program online (http://www.fda.gov/Safety/MedWatch) or by phone (1-800-332-1088).
What should I know about STORAGE and DISPOSAL of this medication?
Keep this medication in the container it came in, tightly closed, and out of reach of children. Store it at room temperature and away from excess heat and moisture (not in the bathroom). Keep the three desiccant (drying agent) pouches in the bottle of medication to keep the tablets dry. Do not eat the desiccant pouches.
It is important to keep all medication out of sight and reach of children as many containers (such as weekly pill minders and those for eye drops, creams, patches, and inhalers) are not child-resistant and young children can open them easily. To protect young children from poisoning, always lock safety caps and immediately place the medication in a safe location – one that is up and away and out of their sight and reach. http://www.upandaway.org
Unneeded medications should be disposed of in special ways to ensure that pets, children, and other people cannot consume them. However, you should not flush this medication down the toilet. Instead, the best way to dispose of your medication is through a medicine take-back program. Talk to your pharmacist or contact your local garbage/recycling department to learn about take-back programs in your community. See the FDA's Safe Disposal of Medicines website (http://goo.gl/c4Rm4p) for more information if you do not have access to a take-back program.
What should I do in case of OVERDOSE?
In case of overdose, call the poison control helpline at 1-800-222-1222. Information is also available online at https://www.poisonhelp.org/help. If the victim has collapsed, had a seizure, has trouble breathing, or can't be awakened, immediately call emergency services at 911.
What OTHER INFORMATION should I know?
Keep all appointments with your doctor and the laboratory. Your doctor may order certain lab tests to check your body's response to etravirine.
Before having any laboratory test, tell your doctor and the laboratory personnel that you are taking etravirine.
Do not let anyone else take your medication. Ask your pharmacist any questions you have about refilling your prescription.
Keep a list of your medications and show it to your doctor and pharmacist when you get a new medication.
It is important for you to keep a written list of all of the prescription and nonprescription (over-the-counter) medicines you are taking, as well as any products such as vitamins, minerals, or other dietary supplements. You should bring this list with you each time you visit a doctor or if you are admitted to a hospital. It is also important information to carry with you in case of emergencies.
Drug interactions
Drug | Interaction |
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Montelukast | Montelukast The metabolism of Montelukast can be decreased when combined with Etravirine. |
Leflunomide | Leflunomide The metabolism of Etravirine can be decreased when combined with Leflunomide. |
Delavirdine | Delavirdine The metabolism of Etravirine can be decreased when combined with Delavirdine. |
Nevirapine | Nevirapine The metabolism of Etravirine can be decreased when combined with Nevirapine. |
Atorvastatin | Atorvastatin The serum concentration of Atorvastatin can be decreased when it is combined with Etravirine. |
Aminophylline | Aminophylline The metabolism of Aminophylline can be increased when combined with Etravirine. |
Candesartan | Candesartan The metabolism of Candesartan can be decreased when combined with Etravirine. |
Cilostazol | Cilostazol The serum concentration of Cilostazol can be increased when it is combined with Etravirine. |
Clopidogrel | Clopidogrel The metabolism of Clopidogrel can be decreased when combined with Etravirine. |
Fenofibrate | Fenofibrate The metabolism of Etravirine can be decreased when combined with Fenofibrate. |
Tacrolimus | Tacrolimus The metabolism of Tacrolimus can be increased when combined with Etravirine. |
Fluconazole Injection | Fluconazole Injection The metabolism of Etravirine can be decreased when combined with Fluconazole. |
Hydromorphone Injection | Hydromorphone Injection The metabolism of Hydromorphone can be decreased when combined with Etravirine. |
Meperidine Injection | Meperidine Injection The metabolism of Meperidine can be increased when combined with Etravirine. |
Metronidazole Injection | Metronidazole Injection The metabolism of Etravirine can be decreased when combined with Metronidazole. |
Zidovudine Injection | Zidovudine Injection The metabolism of Zidovudine can be decreased when combined with Etravirine. |
Cyclosporine | Cyclosporine The metabolism of Cyclosporine can be increased when combined with Etravirine. |
Ondansetron | Ondansetron The metabolism of Ondansetron can be decreased when combined with Etravirine. |
Torsemide | Torsemide The metabolism of Etravirine can be decreased when combined with Torasemide. |
Olanzapine | Olanzapine The metabolism of Etravirine can be decreased when combined with Olanzapine. |
Alosetron | Alosetron The metabolism of Alosetron can be decreased when combined with Etravirine. |
Dofetilide | Dofetilide The metabolism of Dofetilide can be increased when combined with Etravirine. |
Meloxicam | Meloxicam The metabolism of Meloxicam can be decreased when combined with Etravirine. |
Oxcarbazepine | Oxcarbazepine The metabolism of Etravirine can be decreased when combined with Oxcarbazepine. |
Pantoprazole | Pantoprazole The metabolism of Etravirine can be decreased when combined with Pantoprazole. |
Telmisartan | Telmisartan The metabolism of Etravirine can be decreased when combined with Telmisartan. |
Anakinra | Anakinra The metabolism of Etravirine can be increased when combined with Anakinra. |
Trimipramine | Trimipramine The serum concentration of Trimipramine can be decreased when it is combined with Etravirine. |
Etanercept Injection | Etanercept Injection The metabolism of Etravirine can be increased when combined with Etanercept. |
Modafinil | Modafinil The metabolism of Etravirine can be decreased when combined with Modafinil. |
Tenofovir | Tenofovir The metabolism of Tenofovir can be increased when combined with Etravirine. |
Sirolimus | Sirolimus The metabolism of Sirolimus can be increased when combined with Etravirine. |
Epinephrine Injection | Epinephrine Injection The metabolism of Etravirine can be decreased when combined with Epinephrine. |
Escitalopram | Escitalopram The metabolism of Escitalopram can be decreased when combined with Etravirine. |
Zonisamide | Zonisamide The metabolism of Zonisamide can be decreased when combined with Etravirine. |
Adalimumab Injection | Adalimumab Injection The metabolism of Etravirine can be increased when combined with Adalimumab. |
Aripiprazole | Aripiprazole The metabolism of Aripiprazole can be increased when combined with Etravirine. |
Atazanavir | Atazanavir The serum concentration of Etravirine can be increased when it is combined with Atazanavir. |
Eletriptan | Eletriptan The metabolism of Eletriptan can be decreased when combined with Etravirine. |
Rosuvastatin | Rosuvastatin The metabolism of Rosuvastatin can be increased when combined with Etravirine. |
Aprepitant | Aprepitant The metabolism of Etravirine can be decreased when combined with Aprepitant. |
Memantine | Memantine The metabolism of Etravirine can be decreased when combined with Memantine. |
Fosamprenavir | Fosamprenavir The serum concentration of the active metabolites of Fosamprenavir can be increased when Fosamprenavir is used in combination with Etravirine. |
Progesterone | Progesterone The metabolism of Progesterone can be increased when combined with Etravirine. |
Infliximab Injection | Infliximab Injection The metabolism of Etravirine can be increased when combined with Infliximab. |
Oxandrolone | Oxandrolone The metabolism of Etravirine can be decreased when combined with Oxandrolone. |
Rifaximin | Rifaximin The metabolism of Etravirine can be increased when combined with Rifaximin. |
Duloxetine | Duloxetine The metabolism of Duloxetine can be increased when combined with Etravirine. |
Norethindrone | Norethindrone The metabolism of Norethisterone can be increased when combined with Etravirine. |
Bosentan | Bosentan The metabolism of Bosentan can be decreased when combined with Etravirine. |
Erlotinib | Erlotinib The serum concentration of Erlotinib can be decreased when it is combined with Etravirine. |
Eszopiclone | Eszopiclone The serum concentration of Eszopiclone can be decreased when it is combined with Etravirine. |
Voriconazole | Voriconazole The metabolism of Etravirine can be decreased when combined with Voriconazole. |
Peginterferon Alfa-2b (PEG-Intron) | Peginterferon Alfa-2b (PEG-Intron) The metabolism of Etravirine can be increased when combined with Peginterferon alfa-2b. |
Ramelteon | Ramelteon The metabolism of Ramelteon can be decreased when combined with Etravirine. |
Tipranavir | Tipranavir The serum concentration of Etravirine can be decreased when it is combined with Tipranavir. |
Felbamate | Felbamate The metabolism of Etravirine can be decreased when combined with Felbamate. |
Ranolazine | Ranolazine The metabolism of Ranolazine can be increased when combined with Etravirine. |
Abatacept Injection | Abatacept Injection The metabolism of Etravirine can be increased when combined with Abatacept. |
Imatinib | Imatinib The metabolism of Etravirine can be decreased when combined with Imatinib. |
Gefitinib | Gefitinib The metabolism of Etravirine can be decreased when combined with Gefitinib. |
Paliperidone | Paliperidone The serum concentration of Paliperidone can be decreased when it is combined with Etravirine. |
Bortezomib | Bortezomib The metabolism of Etravirine can be increased when combined with Bortezomib. |
Influenza Vaccine, Live Intranasal | Influenza Vaccine, Live Intranasal The therapeutic efficacy of Typhoid Vaccine Live can be decreased when used in combination with Etravirine. |
Live Shingles (Zoster) Vaccine (ZVL) | Live Shingles (Zoster) Vaccine (ZVL) The therapeutic efficacy of Varicella Zoster Vaccine (Live/attenuated) can be decreased when used in combination with Etravirine. |
Nabilone | Nabilone The metabolism of Etravirine can be decreased when combined with Nabilone. |
Retapamulin | Retapamulin The metabolism of Retapamulin can be increased when combined with Etravirine. |
Sorafenib | Sorafenib The metabolism of Etravirine can be increased when combined with Sorafenib. |
Sunitinib | Sunitinib The metabolism of Sunitinib can be increased when combined with Etravirine. |
Dronabinol | Dronabinol The metabolism of Dronabinol can be decreased when combined with Etravirine. |
Lapatinib | Lapatinib The metabolism of Lapatinib can be decreased when combined with Etravirine. |
Dasatinib | Dasatinib The metabolism of Dasatinib can be increased when combined with Etravirine. |
Armodafinil | Armodafinil The metabolism of Etravirine can be decreased when combined with Armodafinil. |
Temsirolimus | Temsirolimus The metabolism of Temsirolimus can be increased when combined with Etravirine. |
Nilotinib | Nilotinib The metabolism of Etravirine can be increased when combined with Nilotinib. |
Bexarotene | Bexarotene The metabolism of Bexarotene can be decreased when combined with Etravirine. |
Chloramphenicol Injection | Chloramphenicol Injection The metabolism of Etravirine can be decreased when combined with Chloramphenicol. |
Nebivolol | Nebivolol The metabolism of Nebivolol can be decreased when combined with Etravirine. |
Tretinoin | Tretinoin The metabolism of Tretinoin can be decreased when combined with Etravirine. |
Bendamustine Injection | Bendamustine Injection The serum concentration of Bendamustine can be decreased when it is combined with Etravirine. |
Flecainide | Flecainide The metabolism of Etravirine can be decreased when combined with Flecainide. |
Certolizumab Injection | Certolizumab Injection The metabolism of Etravirine can be increased when combined with Certolizumab pegol. |
Ixabepilone Injection | Ixabepilone Injection The metabolism of Ixabepilone can be increased when combined with Etravirine. |
Irinotecan Injection | Irinotecan Injection The metabolism of Irinotecan can be increased when combined with Etravirine. |
Praziquantel | Praziquantel The metabolism of Praziquantel can be decreased when combined with Etravirine. |
Rufinamide | Rufinamide The metabolism of Rufinamide can be increased when combined with Etravirine. |
Milnacipran | Milnacipran The metabolism of Milnacipran can be increased when combined with Etravirine. |
Dexlansoprazole | Dexlansoprazole The metabolism of Dexlansoprazole can be decreased when combined with Etravirine. |
Prasugrel | Prasugrel The metabolism of Prasugrel can be decreased when combined with Etravirine. |
Lacosamide | Lacosamide The metabolism of Lacosamide can be decreased when combined with Etravirine. |
Everolimus | Everolimus The metabolism of Everolimus can be increased when combined with Etravirine. |
Tolvaptan (low blood sodium) | Tolvaptan (low blood sodium) The serum concentration of Tolvaptan can be decreased when it is combined with Etravirine. |
Dronedarone | Dronedarone The metabolism of Dronedarone can be increased when combined with Etravirine. |
Romidepsin Injection | Romidepsin Injection The serum concentration of Romidepsin can be decreased when it is combined with Etravirine. |
Tapentadol | Tapentadol The metabolism of Tapentadol can be decreased when combined with Etravirine. |
Topotecan | Topotecan The serum concentration of Topotecan can be decreased when it is combined with Etravirine. |
Golimumab Injection | Golimumab Injection The metabolism of Etravirine can be increased when combined with Golimumab. |
Pazopanib | Pazopanib The metabolism of Pazopanib can be increased when combined with Etravirine. |
Pitavastatin | Pitavastatin The metabolism of Pitavastatin can be decreased when combined with Etravirine. |
Albendazole | Albendazole The metabolism of Albendazole can be decreased when combined with Etravirine. |
Ulipristal | Ulipristal The metabolism of Ulipristal can be increased when combined with Etravirine. |
Levonorgestrel | Levonorgestrel The metabolism of Levonorgestrel can be increased when combined with Etravirine. |
Tocilizumab Injection | Tocilizumab Injection The metabolism of Etravirine can be increased when combined with Tocilizumab. |
Cabazitaxel Injection | Cabazitaxel Injection The serum concentration of Cabazitaxel can be decreased when it is combined with Etravirine. |
Vilazodone | Vilazodone The metabolism of Vilazodone can be decreased when combined with Etravirine. |
Busulfan Injection | Busulfan Injection The metabolism of Busulfan can be increased when combined with Etravirine. |
Roflumilast | Roflumilast The metabolism of Roflumilast can be increased when combined with Etravirine. |
Linagliptin | Linagliptin The serum concentration of Linagliptin can be decreased when it is combined with Etravirine. |
Cyclophosphamide Injection | Cyclophosphamide Injection The metabolism of Cyclophosphamide can be increased when combined with Etravirine. |
Abiraterone | Abiraterone The metabolism of Etravirine can be decreased when combined with Abiraterone. |
Ticagrelor | Ticagrelor The metabolism of Etravirine can be decreased when combined with Ticagrelor. |
Brentuximab Vedotin Injection | Brentuximab Vedotin Injection The serum concentration of Brentuximab vedotin can be decreased when it is combined with Etravirine. |
Ruxolitinib | Ruxolitinib The metabolism of Ruxolitinib can be increased when combined with Etravirine. |
Vandetanib | Vandetanib The metabolism of Vandetanib can be increased when combined with Etravirine. |
Clobazam | Clobazam The metabolism of Clobazam can be decreased when combined with Etravirine. |
Vemurafenib | Vemurafenib The metabolism of Etravirine can be increased when combined with Vemurafenib. |
Vismodegib | Vismodegib The metabolism of Etravirine can be decreased when combined with Vismodegib. |
Axitinib | Axitinib The metabolism of Axitinib can be increased when combined with Etravirine. |
Crizotinib | Crizotinib The metabolism of Crizotinib can be increased when combined with Etravirine. |
Cabergoline | Cabergoline The metabolism of Cabergoline can be increased when combined with Etravirine. |
Carfilzomib Injection | Carfilzomib Injection The serum concentration of Carfilzomib can be decreased when it is combined with Etravirine. |
Enzalutamide | Enzalutamide The metabolism of Etravirine can be increased when combined with Enzalutamide. |
Regorafenib | Regorafenib The serum concentration of Etravirine can be decreased when it is combined with Regorafenib. |
Bosutinib | Bosutinib The metabolism of Bosutinib can be increased when combined with Etravirine. |
Cabozantinib (thyroid cancer) | Cabozantinib (thyroid cancer) The metabolism of Cabozantinib can be decreased when combined with Etravirine. |
Ponatinib | Ponatinib The metabolism of Ponatinib can be increased when combined with Etravirine. |
Pomalidomide | Pomalidomide The serum concentration of Pomalidomide can be decreased when it is combined with Etravirine. |
Ado-trastuzumab Emtansine Injection | Ado-trastuzumab Emtansine Injection The serum concentration of Trastuzumab emtansine can be decreased when it is combined with Etravirine. |
Apixaban | Apixaban The metabolism of Apixaban can be decreased when combined with Etravirine. |
Dabrafenib | Dabrafenib The serum concentration of Etravirine can be decreased when it is combined with Dabrafenib. |
Ospemifene | Ospemifene The metabolism of Ospemifene can be decreased when combined with Etravirine. |
Dolutegravir | Dolutegravir The serum concentration of Dolutegravir can be decreased when it is combined with Etravirine. |
Afatinib | Afatinib The serum concentration of Afatinib can be decreased when it is combined with Etravirine. |
Levomilnacipran | Levomilnacipran The metabolism of Levomilnacipran can be increased when combined with Etravirine. |
Vortioxetine | Vortioxetine The metabolism of Vortioxetine can be decreased when combined with Etravirine. |
Perampanel | Perampanel The metabolism of Perampanel can be increased when combined with Etravirine. |
Lomitapide | Lomitapide The metabolism of Lomitapide can be increased when combined with Etravirine. |
Ketorolac Injection | Ketorolac Injection The metabolism of Ketorolac can be decreased when combined with Etravirine. |
Sofosbuvir | Sofosbuvir The serum concentration of Sofosbuvir can be decreased when it is combined with Etravirine. |
Dapagliflozin | Dapagliflozin The metabolism of Dapagliflozin can be decreased when combined with Etravirine. |
Apremilast | Apremilast The metabolism of Etravirine can be increased when combined with Apremilast. |
Ceritinib | Ceritinib The metabolism of Ceritinib can be increased when combined with Etravirine. |
Siltuximab Injection | Siltuximab Injection The metabolism of Etravirine can be increased when combined with Siltuximab. |
Eslicarbazepine | Eslicarbazepine The metabolism of Etravirine can be decreased when combined with Eslicarbazepine. |
Idelalisib | Idelalisib The metabolism of Idelalisib can be increased when combined with Etravirine. |
Testosterone Injection | Testosterone Injection The metabolism of Testosterone can be decreased when combined with Etravirine. |
Oritavancin Injection | Oritavancin Injection The metabolism of Etravirine can be decreased when combined with Oritavancin. |
Vorapaxar | Vorapaxar The metabolism of Vorapaxar can be increased when combined with Etravirine. |
Suvorexant | Suvorexant The metabolism of Suvorexant can be increased when combined with Etravirine. |
Olaparib | Olaparib The metabolism of Olaparib can be increased when combined with Etravirine. |
Tasimelteon | Tasimelteon The metabolism of Tasimelteon can be increased when combined with Etravirine. |
Nintedanib | Nintedanib The metabolism of Nintedanib can be increased when combined with Etravirine. |
Secukinumab Injection | Secukinumab Injection The metabolism of Etravirine can be increased when combined with Secukinumab. |
Palbociclib | Palbociclib The metabolism of Palbociclib can be increased when combined with Etravirine. |
Lenvatinib | Lenvatinib The metabolism of Etravirine can be decreased when combined with Lenvatinib. |
Naloxegol | Naloxegol The metabolism of Etravirine can be decreased when combined with Naloxegol. |
Panobinostat | Panobinostat The metabolism of Panobinostat can be increased when combined with Etravirine. |
Haloperidol Injection | Haloperidol Injection The serum concentration of Haloperidol can be increased when it is combined with Etravirine. |
Sonidegib | Sonidegib The metabolism of Sonidegib can be increased when combined with Etravirine. |
Rolapitant | Rolapitant The metabolism of Rolapitant can be increased when combined with Etravirine. |
Daclatasvir | Daclatasvir The metabolism of Daclatasvir can be increased when combined with Etravirine. |
Ziprasidone Injection | Ziprasidone Injection The metabolism of Ziprasidone can be increased when combined with Etravirine. |
Cobimetinib | Cobimetinib The metabolism of Cobimetinib can be increased when combined with Etravirine. |
Trabectedin Injection | Trabectedin Injection The metabolism of Trabectedin can be increased when combined with Etravirine. |
Osimertinib | Osimertinib The serum concentration of Osimertinib can be decreased when it is combined with Etravirine. |
Alectinib | Alectinib The metabolism of Alectinib can be increased when combined with Etravirine. |
Ixazomib | Ixazomib The metabolism of Ixazomib can be increased when combined with Etravirine. |
Rifapentine | Rifapentine The metabolism of Etravirine can be increased when combined with Rifapentine. |
Lesinurad | Lesinurad The metabolism of Lesinurad can be decreased when combined with Etravirine. |
Brivaracetam Injection | Brivaracetam Injection The metabolism of Brivaracetam can be decreased when combined with Etravirine. |
Venetoclax | Venetoclax The metabolism of Venetoclax can be increased when combined with Etravirine. |
Diphenhydramine Injection | Diphenhydramine Injection The metabolism of Diphenhydramine can be decreased when combined with Etravirine. |
Rucaparib | Rucaparib The metabolism of Etravirine can be decreased when combined with Rucaparib. |
Ribociclib | Ribociclib The metabolism of Etravirine can be increased when combined with Ribociclib. |
Brigatinib | Brigatinib The metabolism of Brigatinib can be increased when combined with Etravirine. |
Doxepin (Insomnia) | Doxepin (Insomnia) The metabolism of Doxepin can be decreased when combined with Etravirine. |
Deflazacort | Deflazacort The serum concentration of Deflazacort can be decreased when it is combined with Etravirine. |
Safinamide | Safinamide The metabolism of Etravirine can be decreased when combined with Safinamide. |
Midostaurin | Midostaurin The metabolism of Etravirine can be increased when combined with Midostaurin. |
Neratinib | Neratinib The metabolism of Neratinib can be increased when combined with Etravirine. |
Enasidenib | Enasidenib The metabolism of Etravirine can be increased when combined with Enasidenib. |
Inotuzumab Ozogamicin Injection | Inotuzumab Ozogamicin Injection The serum concentration of Inotuzumab ozogamicin can be decreased when it is combined with Etravirine. |
Aprepitant/Fosaprepitant Injection | Aprepitant/Fosaprepitant Injection The metabolism of Fosaprepitant can be increased when combined with Etravirine. |
Copanlisib Injection | Copanlisib Injection The metabolism of Copanlisib can be increased when combined with Etravirine. |
Delafloxacin | Delafloxacin The metabolism of Etravirine can be increased when combined with Delafloxacin. |
Abemaciclib | Abemaciclib The metabolism of Abemaciclib can be increased when combined with Etravirine. |
Acalabrutinib | Acalabrutinib The metabolism of Acalabrutinib can be increased when combined with Etravirine. |
Letermovir | Letermovir The metabolism of Etravirine can be increased when combined with Letermovir. |
Buprenorphine Injection | Buprenorphine Injection The metabolism of Etravirine can be decreased when combined with Buprenorphine. |
Apalutamide | Apalutamide The serum concentration of Etravirine can be increased when it is combined with Apalutamide. |
Avatrombopag | Avatrombopag The metabolism of Etravirine can be increased when combined with Avatrombopag. |
Baricitinib | Baricitinib The metabolism of Baricitinib can be increased when combined with Etravirine. |
Binimetinib | Binimetinib The serum concentration of Binimetinib can be decreased when it is combined with Etravirine. |
Ivosidenib | Ivosidenib The metabolism of Ivosidenib can be increased when combined with Etravirine. |
Cannabidiol | Cannabidiol The metabolism of Cannabidiol can be decreased when combined with Etravirine. |
Dacomitinib | Dacomitinib The metabolism of Dacomitinib can be increased when combined with Etravirine. |
Duvelisib | Duvelisib The metabolism of Duvelisib can be increased when combined with Etravirine. |
Stiripentol | Stiripentol The metabolism of Etravirine can be decreased when combined with Stiripentol. |
Talazoparib | Talazoparib The serum concentration of Talazoparib can be decreased when it is combined with Etravirine. |
Gilteritinib | Gilteritinib The metabolism of Gilteritinib can be increased when combined with Etravirine. |
Lorlatinib | Lorlatinib The metabolism of Lorlatinib can be decreased when combined with Etravirine. |
Paclitaxel (with albumin) Injection | Paclitaxel (with albumin) Injection The metabolism of Paclitaxel can be increased when combined with Etravirine. |
Rifamycin | Rifamycin The metabolism of Etravirine can be increased when combined with Rifamycin. |
Prucalopride | Prucalopride The metabolism of Prucalopride can be increased when combined with Etravirine. |
Emapalumab-lzsg Injection | Emapalumab-lzsg Injection The metabolism of Etravirine can be increased when combined with Emapalumab. |
Siponimod | Siponimod The metabolism of Siponimod can be increased when combined with Etravirine. |
Erdafitinib | Erdafitinib The metabolism of Erdafitinib can be increased when combined with Etravirine. |
Esomeprazole Injection | Esomeprazole Injection The metabolism of Etravirine can be decreased when combined with Esomeprazole. |
Alpelisib | Alpelisib The serum concentration of Etravirine can be decreased when it is combined with Alpelisib. |
Darolutamide | Darolutamide The serum concentration of Darolutamide can be decreased when it is combined with Etravirine. |
Triclabendazole | Triclabendazole The metabolism of Etravirine can be decreased when combined with Triclabendazole. |
Entrectinib | Entrectinib The metabolism of Entrectinib can be increased when combined with Etravirine. |
Pexidartinib | Pexidartinib The metabolism of Pexidartinib can be increased when combined with Etravirine. |
Istradefylline | Istradefylline The metabolism of Istradefylline can be decreased when combined with Etravirine. |
Pitolisant | Pitolisant The serum concentration of Etravirine can be decreased when it is combined with Pitolisant. |
Fedratinib | Fedratinib The metabolism of Fedratinib can be decreased when combined with Etravirine. |
Lefamulin | Lefamulin The metabolism of Lefamulin can be increased when combined with Etravirine. |
Phenytoin Injection | Phenytoin Injection The serum concentration of Etravirine can be decreased when it is combined with Phenytoin. |
Fosphenytoin Injection | Fosphenytoin Injection The serum concentration of Etravirine can be decreased when it is combined with Fosphenytoin. |
Zanubrutinib | Zanubrutinib The metabolism of Zanubrutinib can be increased when combined with Etravirine. |
Voxelotor | Voxelotor The serum concentration of Voxelotor can be decreased when it is combined with Etravirine. |
Avapritinib | Avapritinib The metabolism of Avapritinib can be decreased when combined with Etravirine. |
Lumateperone | Lumateperone The serum concentration of Lumateperone can be decreased when it is combined with Etravirine. |
Ubrogepant | Ubrogepant The serum concentration of Ubrogepant can be decreased when it is combined with Etravirine. |
Tazemetostat | Tazemetostat The metabolism of Tazemetostat can be increased when combined with Etravirine. |
Cenobamate | Cenobamate The serum concentration of Etravirine can be decreased when it is combined with Cenobamate. |
Pemigatinib | Pemigatinib The metabolism of Pemigatinib can be increased when combined with Etravirine. |
Selumetinib | Selumetinib The serum concentration of Selumetinib can be decreased when it is combined with Etravirine. |
Rimegepant | Rimegepant The metabolism of Rimegepant can be increased when combined with Etravirine. |
Tucatinib | Tucatinib The metabolism of Tucatinib can be decreased when combined with Etravirine. |
Selpercatinib | Selpercatinib The serum concentration of Selpercatinib can be decreased when it is combined with Etravirine. |
Capmatinib | Capmatinib The serum concentration of Capmatinib can be decreased when it is combined with Etravirine. |
Lemborexant | Lemborexant The serum concentration of Lemborexant can be decreased when it is combined with Etravirine. |
Lurbinectedin Injection | Lurbinectedin Injection The serum concentration of Lurbinectedin can be decreased when it is combined with Etravirine. |
Pralsetinib | Pralsetinib The metabolism of Etravirine can be decreased when combined with Pralsetinib. |
Satralizumab-mwge Injection | Satralizumab-mwge Injection The serum concentration of Etravirine can be decreased when it is combined with Satralizumab. |
Relugolix | Relugolix The serum concentration of Relugolix can be decreased when it is combined with Etravirine. |
Progestin-Only (drospirenone) Oral Contraceptives | Progestin-Only (drospirenone) Oral Contraceptives The metabolism of Drospirenone can be increased when combined with Etravirine. |
Theophylline | Theophylline The metabolism of Theophylline can be increased when combined with Etravirine. |
Indomethacin | Indomethacin The metabolism of Indomethacin can be decreased when combined with Etravirine. |
Mefenamic Acid | Mefenamic Acid The metabolism of Mefenamic acid can be decreased when combined with Etravirine. |
Naproxen | Naproxen The metabolism of Naproxen can be decreased when combined with Etravirine. |
Floxuridine | Floxuridine The metabolism of Etravirine can be decreased when combined with Floxuridine. |
Phenobarbital | Phenobarbital The metabolism of Etravirine can be increased when combined with Phenobarbital. |
Methotrexate Injection | Methotrexate Injection The metabolism of Methotrexate can be increased when combined with Etravirine. |
Primidone | Primidone The metabolism of Etravirine can be increased when combined with Primidone. |
Methsuximide | Methsuximide The metabolism of Etravirine can be decreased when combined with Methsuximide. |
Chlorpromazine | Chlorpromazine The metabolism of Chlorpromazine can be increased when combined with Etravirine. |
Diazepam | Diazepam The metabolism of Diazepam can be decreased when combined with Etravirine. |
Lorazepam | Lorazepam The metabolism of Lorazepam can be increased when combined with Etravirine. |
Tranylcypromine | Tranylcypromine The metabolism of Etravirine can be decreased when combined with Tranylcypromine. |
Phenelzine | Phenelzine The metabolism of Etravirine can be decreased when combined with Phenelzine. |
Prochlorperazine | Prochlorperazine The metabolism of Prochlorperazine can be increased when combined with Etravirine. |
Thioridazine | Thioridazine The metabolism of Thioridazine can be decreased when combined with Etravirine. |
Dapsone | Dapsone The metabolism of Dapsone can be decreased when combined with Etravirine. |
Sulfadiazine | Sulfadiazine The metabolism of Etravirine can be decreased when combined with Sulfadiazine. |
Methadone | Methadone The metabolism of Methadone can be decreased when combined with Etravirine. |
Ibuprofen | Ibuprofen The metabolism of Ibuprofen can be decreased when combined with Etravirine. |
Phentermine | Phentermine The metabolism of Phentermine can be increased when combined with Etravirine. |
Doxorubicin | Doxorubicin The serum concentration of Doxorubicin can be decreased when it is combined with Etravirine. |
Dactinomycin | Dactinomycin The serum concentration of Dactinomycin can be decreased when it is combined with Etravirine. |
Carbamazepine | Carbamazepine The metabolism of Carbamazepine can be increased when combined with Etravirine. |
Clonidine | Clonidine The metabolism of Clonidine can be increased when combined with Etravirine. |
Cimetidine | Cimetidine The metabolism of Etravirine can be decreased when combined with Cimetidine. |
Warfarin | Warfarin The metabolism of Warfarin can be increased when combined with Etravirine. |
Clonazepam | Clonazepam The metabolism of Clonazepam can be increased when combined with Etravirine. |
Promethazine | Promethazine The metabolism of Etravirine can be decreased when combined with Promethazine. |
Digoxin | Digoxin The serum concentration of Digoxin can be increased when it is combined with Etravirine. |
Quinine | Quinine The metabolism of Etravirine can be decreased when combined with Quinine. |
Sulfinpyrazone | Sulfinpyrazone The metabolism of Etravirine can be decreased when combined with Sulfinpyrazone. |
Isosorbide | Isosorbide The metabolism of Isosorbide can be increased when combined with Etravirine. |
Clindamycin Injection | Clindamycin Injection The metabolism of Clindamycin can be increased when combined with Etravirine. |
Amitriptyline | Amitriptyline The metabolism of Amitriptyline can be decreased when combined with Etravirine. |
Imipramine | Imipramine The serum concentration of Etravirine can be decreased when it is combined with Imipramine. |
Probenecid | Probenecid The metabolism of Etravirine can be decreased when combined with Probenecid. |
Quinidine | Quinidine The metabolism of Quinidine can be increased when combined with Etravirine. |
Isoniazid | Isoniazid The metabolism of Etravirine can be decreased when combined with Isoniazid. |
Rifampin | Rifampin The metabolism of Etravirine can be increased when combined with Rifampicin. |
Valproic Acid | Valproic Acid The metabolism of Etravirine can be decreased when combined with Valproic acid. |
Tamoxifen | Tamoxifen The metabolism of Tamoxifen can be increased when combined with Etravirine. |
Methimazole | Methimazole The metabolism of Etravirine can be decreased when combined with Methimazole. |
Chlorpropamide | Chlorpropamide The metabolism of Chlorpropamide can be decreased when combined with Etravirine. |
Tolbutamide | Tolbutamide The metabolism of Tolbutamide can be decreased when combined with Etravirine. |
Tolazamide | Tolazamide The metabolism of Tolazamide can be decreased when combined with Etravirine. |
Dextromethorphan | Dextromethorphan The metabolism of Dextromethorphan can be decreased when combined with Etravirine. |
Carisoprodol | Carisoprodol The metabolism of Carisoprodol can be decreased when combined with Etravirine. |
Propranolol (Cardiovascular) | Propranolol (Cardiovascular) The serum concentration of Propranolol can be increased when it is combined with Etravirine. |
Nortriptyline | Nortriptyline The serum concentration of Nortriptyline can be decreased when it is combined with Etravirine. |
Fluorouracil Injection | Fluorouracil Injection The metabolism of Etravirine can be decreased when combined with Fluorouracil. |
Cephalexin | Cephalexin The metabolism of Cephalexin can be increased when combined with Etravirine. |
Bacillus Calmette-Guerin (BCG) Vaccine | Bacillus Calmette-Guerin (BCG) Vaccine The therapeutic efficacy of Bacillus calmette-guerin substrain tice live antigen can be decreased when used in combination with Etravirine. |
Ketoconazole | Ketoconazole The metabolism of Etravirine can be decreased when combined with Ketoconazole. |
Thiotepa Injection | Thiotepa Injection The metabolism of Thiotepa can be increased when combined with Etravirine. |
Vincristine Injection | Vincristine Injection The serum concentration of Vincristine can be decreased when it is combined with Etravirine. |
Vinblastine | Vinblastine The metabolism of Vinblastine can be increased when combined with Etravirine. |
Metoprolol | Metoprolol The metabolism of Metoprolol can be increased when combined with Etravirine. |
Aspirin | Aspirin The metabolism of Acetylsalicylic acid can be decreased when combined with Etravirine. |
Trimethoprim | Trimethoprim The metabolism of Trimethoprim can be decreased when combined with Etravirine. |
Diltiazem | Diltiazem The metabolism of Diltiazem can be decreased when combined with Etravirine. |
Timolol | Timolol The metabolism of Timolol can be decreased when combined with Etravirine. |
Verapamil | Verapamil The metabolism of Etravirine can be decreased when combined with Verapamil. |
Cisplatin Injection | Cisplatin Injection The metabolism of Etravirine can be decreased when combined with Cisplatin. |
Piroxicam | Piroxicam The metabolism of Piroxicam can be decreased when combined with Etravirine. |
Etoposide | Etoposide The metabolism of Etoposide can be increased when combined with Etravirine. |
Glyburide | Glyburide The metabolism of Etravirine can be decreased when combined with Glyburide. |
Glipizide | Glipizide The metabolism of Glipizide can be decreased when combined with Etravirine. |
Labetalol | Labetalol The metabolism of Labetalol can be decreased when combined with Etravirine. |
Gemfibrozil | Gemfibrozil The metabolism of Etravirine can be decreased when combined with Gemfibrozil. |
Pimozide | Pimozide The metabolism of Pimozide can be increased when combined with Etravirine. |
Flurbiprofen | Flurbiprofen The metabolism of Flurbiprofen can be decreased when combined with Etravirine. |
Amiodarone | Amiodarone The metabolism of Amiodarone can be increased when combined with Etravirine. |
Lovastatin | Lovastatin The serum concentration of Lovastatin can be decreased when it is combined with Etravirine. |
Diclofenac | Diclofenac The metabolism of Diclofenac can be decreased when combined with Etravirine. |
Fluoxetine | Fluoxetine The metabolism of Etravirine can be decreased when combined with Fluoxetine. |
Clozapine | Clozapine The metabolism of Etravirine can be decreased when combined with Clozapine. |
Idarubicin | Idarubicin The metabolism of Idarubicin can be decreased when combined with Etravirine. |
Etodolac | Etodolac The metabolism of Etodolac can be decreased when combined with Etravirine. |
Felodipine | Felodipine The metabolism of Etravirine can be decreased when combined with Felodipine. |
Nabumetone | Nabumetone The metabolism of Nabumetone can be decreased when combined with Etravirine. |
Simvastatin | Simvastatin The serum concentration of Simvastatin can be decreased when it is combined with Etravirine. |
Teniposide Injection | Teniposide Injection The metabolism of Etravirine can be increased when combined with Teniposide. |
Atovaquone | Atovaquone The metabolism of Etravirine can be decreased when combined with Atovaquone. |
Rifabutin | Rifabutin The serum concentration of Etravirine can be decreased when it is combined with Rifabutin. |
Zolpidem | Zolpidem The metabolism of Zolpidem can be decreased when combined with Etravirine. |
Doxazosin | Doxazosin The metabolism of Doxazosin can be increased when combined with Etravirine. |
Omeprazole | Omeprazole The metabolism of Etravirine can be decreased when combined with Omeprazole. |
Cisapride | Cisapride The metabolism of Cisapride can be increased when combined with Etravirine. |
Fluvastatin | Fluvastatin The serum concentration of Fluvastatin can be increased when it is combined with Etravirine. |
Venlafaxine | Venlafaxine The metabolism of Venlafaxine can be decreased when combined with Etravirine. |
Famciclovir | Famciclovir The metabolism of Famciclovir can be increased when combined with Etravirine. |
Fluvoxamine | Fluvoxamine The metabolism of Etravirine can be decreased when combined with Fluvoxamine. |
Losartan | Losartan The metabolism of Etravirine can be decreased when combined with Losartan. |
Tramadol | Tramadol The metabolism of Tramadol can be increased when combined with Etravirine. |
Vinorelbine Injection | Vinorelbine Injection The metabolism of Vinorelbine can be increased when combined with Etravirine. |
Lansoprazole | Lansoprazole The metabolism of Etravirine can be decreased when combined with Lansoprazole. |
Ifosfamide Injection | Ifosfamide Injection The metabolism of Ifosfamide can be increased when combined with Etravirine. |
Nicardipine | Nicardipine The metabolism of Etravirine can be decreased when combined with Nicardipine. |
Bupropion | Bupropion The metabolism of Bupropion can be decreased when combined with Etravirine. |
Ticlopidine | Ticlopidine The metabolism of Etravirine can be decreased when combined with Ticlopidine. |
Glimepiride | Glimepiride The metabolism of Glimepiride can be decreased when combined with Etravirine. |
Gemcitabine Injection | Gemcitabine Injection The serum concentration of Gemcitabine can be decreased when it is combined with Etravirine. |
Ritonavir | Ritonavir The serum concentration of Etravirine can be decreased when it is combined with Ritonavir. |
Docetaxel Injection | Docetaxel Injection The metabolism of Docetaxel can be increased when combined with Etravirine. |
Clomipramine | Clomipramine The metabolism of Etravirine can be increased when combined with Clomipramine. |
Zafirlukast | Zafirlukast The metabolism of Etravirine can be decreased when combined with Zafirlukast. |
Topiramate | Topiramate The metabolism of Topiramate can be decreased when combined with Etravirine. |
Zileuton | Zileuton The metabolism of Zileuton can be decreased when combined with Etravirine. |
Valsartan | Valsartan The metabolism of Etravirine can be decreased when combined with Valsartan. |
Donepezil | Donepezil The metabolism of Donepezil can be decreased when combined with Etravirine. |
Nelfinavir | Nelfinavir The metabolism of Etravirine can be decreased when combined with Nelfinavir. |
Azithromycin | Azithromycin The metabolism of Azithromycin can be increased when combined with Etravirine. |
Carvedilol | Carvedilol The metabolism of Carvedilol can be decreased when combined with Etravirine. |
Nilutamide | Nilutamide The metabolism of Etravirine can be decreased when combined with Nilutamide. |
Selegiline | Selegiline The metabolism of Selegiline can be decreased when combined with Etravirine. |
Bicalutamide | Bicalutamide The metabolism of Etravirine can be increased when combined with Bicalutamide. |
Sertraline | Sertraline The metabolism of Etravirine can be decreased when combined with Sertraline. |
Letrozole | Letrozole The metabolism of Etravirine can be decreased when combined with Letrozole. |
Irbesartan | Irbesartan The metabolism of Irbesartan can be decreased when combined with Etravirine. |
Paroxetine | Paroxetine The metabolism of Etravirine can be decreased when combined with Paroxetine. |
Tolcapone | Tolcapone The metabolism of Etravirine can be decreased when combined with Tolcapone. |
Citalopram | Citalopram Etravirine may increase the QTc-prolonging activities of Citalopram. |
Capecitabine | Capecitabine The metabolism of Etravirine can be decreased when combined with Capecitabine. |
Efavirenz | Efavirenz The metabolism of Etravirine can be decreased when combined with Efavirenz. |
Sildenafil | Sildenafil The metabolism of Sildenafil can be decreased when combined with Etravirine. |
Celecoxib | Celecoxib The metabolism of Celecoxib can be decreased when combined with Etravirine. |
Rosiglitazone | Rosiglitazone The metabolism of Rosiglitazone can be decreased when combined with Etravirine. |
Tolterodine | Tolterodine The metabolism of Tolterodine can be decreased when combined with Etravirine. |
Thalidomide | Thalidomide The metabolism of Etravirine can be decreased when combined with Thalidomide. |
Nateglinide | Nateglinide The metabolism of Nateglinide can be decreased when combined with Etravirine. |
Rabeprazole | Rabeprazole The metabolism of Etravirine can be decreased when combined with Rabeprazole. |
Terbinafine | Terbinafine The metabolism of Terbinafine can be decreased when combined with Etravirine. |
Content provided by: AHFS® Patient Medication Information™. © Copyright, 2021. The American Society of Health-System Pharmacists