FDA-filed SPL labeling · retrieved through openFDA

Gatifloxacin Ophthalmic

Gatifloxacin ophthalmic is an antibiotic eye drop used to treat bacterial conjunctivitis (pink eye).

Brand names ZymaxidZymar
Drug classes ⓘ Quinolone Antimicrobial
Rx Form 1 Route Ophthalmic
Dr. Brian Staiger, PharmD, BCPS
Reviewed by Last reviewed Jul 10, 2026
🧬 Where this information comes from Click to expand

The clinical label records used on this page are FDA-filed Structured Product Labeling (SPL) retrieved through openFDA. We identified 5 clinical label sets within the page’s selected clinical scope after exact ingredient or ingredient-combination matching and applicable route/form matching. Forms, routes, brands, labelers, strengths, and NDC product-record counts are built separately from matching FDA National Drug Code Directory records. The linked DailyMed document is a representative official source for verification, not the page’s only clinical source. View the linked label on DailyMed →

At a glance
Linked label effectiveSep 8, 2016
Clinical labels in scope ⓘ5
AvailabilityRx
Earliest approval/marketing year ⓘ2003
FDA-listed product records ⓘ12
Boxed warningNone found in compared labels
How we combine label and product data →
✓No current FDA shortage listed · checked Sep 26, 2026
⭐ Gatifloxacin Ophthalmic at a glance The quick version — the full detail is in the Patient Information Guide below.
💊
HelloPharmacist Editorial Team Bottom Line
Gatifloxacin ophthalmic solution 0.5% (Zymaxid) is an antibiotic eye drop that effectively treats bacterial conjunctivitis when used as directed for the full 7-day course. Serious allergic reactions are rare but can happen fast — stop the drops and seek help immediately if you have trouble breathing, severe swelling, or a serious skin reaction. Always use the drops only in the eye, follow the dosing schedule, and finish the full course even if your eye feels better sooner.

📖 Gatifloxacin Ophthalmic: Patient Information Guide

A plain-language walkthrough of Gatifloxacin Ophthalmic — what it treats, how it works, how it’s taken, side effects, warnings and interactions. Tap any section to expand it.

🎯What it's used for▾

Gatifloxacin ophthalmic solution 0.5% is an antibiotic eye drop approved to treat bacterial conjunctivitis (pink eye) caused by specific susceptible bacteria.

  • Zymaxid (gatifloxacin ophthalmic solution 0.5%) treats bacterial conjunctivitis caused by Staphylococcus aureus
  • Zymaxid treats bacterial conjunctivitis caused by Staphylococcus epidermidis
  • Zymaxid treats bacterial conjunctivitis caused by Streptococcus mitis group and Streptococcus oralis (studied in fewer than 10 infections each)
  • Zymaxid treats bacterial conjunctivitis caused by Streptococcus pneumoniae
  • Zymaxid treats bacterial conjunctivitis caused by Haemophilus influenzae
  • Zymaxid is approved for use in patients one year of age and older
⚙️How it works▾

Gatifloxacin is a quinolone antibiotic that works by blocking two enzymes bacteria need to survive: DNA gyrase and topoisomerase IV. These enzymes help bacteria copy, repair, and divide their DNA. When gatifloxacin blocks them, the bacteria can no longer replicate and they die. Because it works differently from antibiotic classes like aminoglycosides, macrolides, and tetracyclines, it can sometimes be effective against bacteria resistant to those drugs.

When used as eye drops, blood levels of gatifloxacin remain extremely low — in clinical studies, levels were undetectable in the bloodstream — so the antibiotic effect is largely local, right where it's applied in the eye.

💊How it's taken▾

Zymaxid eye drops follow a two-phase schedule over 7 days. The dosing is more frequent on the first day, then tapers off:

  • Day 1: One drop in the affected eye(s) every two hours while awake, up to 8 times
  • Days 2–7: One drop in the affected eye(s) two to four times daily while awake

Follow your prescriber's exact instructions. Complete the full course of treatment even if your eye starts to feel better early — stopping too soon can allow the infection to return.

🤒Side effects — in detail▾

Most side effects with gatifloxacin eye drops are mild and affect the eyes or mouth. Common ones (reported in 1% or more of patients in clinical studies) include:

  • Worsening of conjunctivitis symptoms
  • Eye irritation
  • Eye pain
  • Dysgeusia — an unusual or bad taste in the mouth
  • Eye discharge, dry eye, or increased tearing
  • Eyelid swelling
  • Headache
  • Reduced visual acuity (blurred or reduced sharpness of vision)

Serious reactions such as severe allergic reactions (including anaphylaxis and throat swelling), difficulty breathing, or signs of Stevens-Johnson Syndrome (severe blistering rash) require immediate medical attention — stop the drops and call for help right away.

⚠️Warnings & precautions▾
  • Serious allergic reactions: Even a single dose can trigger anaphylaxis, severe swelling of the throat or face, difficulty breathing, hives, or — rarely — Stevens-Johnson Syndrome. Stop the medication immediately and seek emergency care if these occur.
  • Superinfection with prolonged use: Using these drops longer than prescribed can allow resistant organisms, including fungi, to grow in the eye. If symptoms worsen or change, contact your doctor.
  • Eye use only: Gatifloxacin ophthalmic solution is strictly for the eye. If it were to enter the front chamber of the eye directly, it could damage the inner lining of the cornea (corneal endothelial cells). Do not attempt to inject or otherwise misuse these drops.
🔀What it interacts with▾

The FDA label for gatifloxacin ophthalmic solution 0.5% does not identify specific drug, food, or substance interactions for this topical eye drop formulation.

    This is not a complete list of interactions. Always talk with your doctor or pharmacist before starting, stopping, or changing any medication.

    📋Before taking it▾
    • Allergy to quinolones: Do not use if you have ever had an allergic reaction to gatifloxacin or any other quinolone antibiotic — this is a contraindication
    • Allergy to ingredients: Tell your doctor if you are allergic to any component of this product
    • Pregnancy: There is no human data on gatifloxacin eye drops in pregnancy; discuss the risks and benefits with your doctor
    • Breastfeeding: It is not known whether this medication reaches breast milk at measurable levels when used as eye drops; discuss with your doctor
    • Infants under 1 year: Safety and effectiveness have not been established in children younger than one year of age
    • Children 1 year and older: Shown to be safe and effective in clinical trials for this age group
    • Older adults: No differences in safety or effectiveness compared to younger adults; no special precautions noted
    🔬Pharmacokinetics — how your body processes it▾

    When gatifloxacin ophthalmic solution 0.5% is applied to the eye, very little of the drug is absorbed into the bloodstream. In a clinical study, blood levels were undetectable (below 5 ng/mL) at all time points — even with intensive dosing of two drops up to 8 times a day. This means the medication works locally in the eye with minimal systemic (whole-body) exposure.

    📦How to store it▾

    Store at 20° to 25°C (68° to 77°F) . Protect from freezing.

    📄 Written from Gatifloxacin Ophthalmic’s FDA-approved label information, summarized in plain language with AI, and reviewed by our pharmacy team before publication. Every point is grounded in that labeling — nothing is invented. How we use AI →

    🩺 Pharmacist Counseling Corner

    Quick, plain-English answers to the questions patients ask most about Gatifloxacin Ophthalmic — the kind of thing our pharmacy team would talk through with you at the counter.

    What exactly is Zymaxid used for? ▾
    Zymaxid is an antibiotic eye drop used to treat bacterial pink eye (bacterial conjunctivitis). It targets specific bacteria that commonly cause eye infections, like Staphylococcus aureus and Streptococcus pneumoniae. It's not for viral pink eye — antibiotics don't work against viruses — so your doctor will confirm the type of infection before prescribing it.
    How do I use the drops, and does the schedule change over time? ▾
    Yes, the schedule is a bit different on the first day. On Day 1, you put one drop in the affected eye every two hours while you're awake, up to 8 times. Starting on Day 2 and through Day 7, you drop back to just two to four drops a day while awake. It's a 7-day course in total — try to finish all 7 days even if your eye feels better after a few days.
    What side effects should I expect, and which ones should make me call the doctor? ▾
    The most common things people notice are mild eye irritation, eye pain, and sometimes a strange taste in the mouth — that last one sounds odd, but it happens with eye drops because of the tear duct connection to the back of the throat. These are usually not serious. What you do need to act on quickly is any sign of a severe allergic reaction: swelling of your face or throat, trouble breathing, hives, or a blistering rash. Those are rare but serious — stop the drops and get medical help right away if that happens.
    Can I use these drops if I'm pregnant or breastfeeding? ▾
    There's no human study data on using gatifloxacin eye drops during pregnancy, so this is definitely a conversation to have with your doctor or OB. The good news is that blood levels from eye drops are essentially undetectable, which means very little of the medication gets into your system — but it's still important to discuss it with your prescriber so they can weigh the benefits and risks for your specific situation.
    My eye is feeling a lot better after 2 days — can I stop the drops early? ▾
    It's tempting to stop when you feel better, but try to finish the full 7-day course. Stopping too soon can leave some bacteria behind, and those survivors can come back — sometimes stronger. Using antibiotics for the full prescribed time is the best way to clear the infection completely and reduce the chance of it returning.
    Is it safe to give these drops to my child? ▾
    Gatifloxacin ophthalmic solution 0.5% has been shown to be safe and effective for children one year of age and older. It has not been studied in babies under 12 months, so it's not recommended for that age group. If your child is over one year old, follow the same dosing schedule as adults and check with your pediatrician if you have any concerns.
    Is Gatifloxacin Ophthalmic available over the counter? ▾
    Gatifloxacin Ophthalmic is dispensed by prescription according to its FDA labeling, so it isn't sold over the counter. Your prescriber and pharmacist will determine if it's appropriate for you.
    When was Gatifloxacin Ophthalmic first available? ▾
    Gatifloxacin Ophthalmic has been available in the United States since at least 2003, based on FDA approval history (Drugs@FDA) and product marketing records.
    Who makes Gatifloxacin Ophthalmic? ▾
    Gatifloxacin Ophthalmic is supplied by 8 manufacturers listed in the FDA NDC Directory, including Allergan, Inc., Pacific Pharma, Inc., Sandoz Inc.

    💬 Answers drafted from Gatifloxacin Ophthalmic’s FDA-approved label information, summarized in plain language with AI, and reviewed by our pharmacy team before publication. Grounded in that labeling — nothing is made up. How we use AI →

    🧰 Keep exploring

    💊 How Gatifloxacin Ophthalmic comes

    Gatifloxacin Ophthalmic is available in 1 form. Different forms and brands can have different approved uses, doses, schedules, and directions. Follow the instructions for your exact product, and do not switch forms without guidance from your prescriber or pharmacist.

    Eye drops

    In the eye
    Brands Zymaxid
    How this form is used
    What it may be used for
    • Zymaxid is used to treat bacterial conjunctivitis (pink eye) caused by susceptible bacteria including Staphylococcus aureus, Staphylococcus epidermidis, Streptococcus pneumoniae, and Haemophilus influenzae
    • Zymaxid has been shown to be safe and effective for bacterial conjunctivitis in patients one year of age and older
    Important instructions
    • Zymaxid: On Day 1, instill one drop into the affected eye(s) every two hours while awake, up to 8 times
    • Zymaxid: On Days 2 through 7, instill one drop two to four times daily in the affected eye(s) while awake
    • Zymaxid is for eye use only — do not swallow or inject
    • Zymaxid: Follow your prescriber's instructions and complete the full 7-day course
    Available strengths 1 strength
    12 FDA-listed product records ⓘ

    📊 Gatifloxacin Ophthalmic across the U.S. market

    How Gatifloxacin Ophthalmic appears in the FDA’s National Drug Code Directory — including its dosage forms, strengths, brand names, manufacturers, and FDA-listed product records. These are directory records, not sales or prescription volume.

    1
    Dose forms ⓘ
    8
    Manufacturers
    3
    Brand names
    12
    FDA-listed product records ⓘ
    2003
    First marketed ⓘ
    Allergan, Inc.25%
    Pacific Pharma, Inc.17%
    Sandoz Inc17%
    Akorn8%
    Caplin Steriles Limited8%
    Leading Pharma, LLC8%
    Other makers17%

    Share of FDA-listed product records by manufacturer — FDA National Drug Code Directory. Record counts are not sales or prescription volume.

    📈 How widely Gatifloxacin Ophthalmic is used

    A general measure of how commonly Gatifloxacin Ophthalmic is prescribed, based on Medicaid — one of the largest public drug programs. The figure below is prescriptions filled in Q1–Q4 2025, summed across every form and brand of the drug.

    Think of this as a proxy for how widely Gatifloxacin Ophthalmic is used, drawn from freely available public data. Medicaid is just one program — these numbers don’t include Medicare, other government coverage, or commercial and cash-pay prescriptions, so real-world use is higher than what’s shown here.

    390
    Medicaid prescriptions filled (Q1–Q4 2025)
    $15,307 gross Medicaid reimbursement (before mandatory rebates — net cost is lower)

    How commonly is Gatifloxacin Ophthalmic prescribed? Of the 1,597 medications we measure, Gatifloxacin Ophthalmic ranks #1,385 by Medicaid prescriptions — more than 13% of them.

    Where Gatifloxacin Ophthalmic ranks among the drugs we measure · Q1–Q4 2025 · neighbors ±5

    Utilization by Gatifloxacin Ophthalmic product

    Pick a product to see its own Medicaid numbers. Each chip is one clinical product — a specific strength & dosage form as defined by RxNorm — with brand-name and generic versions combined.

    gatifloxacin 5 MG/ML Ophthalmic Solution

    390 Medicaid prescriptions (Q1–Q4 2025) 100% of Gatifloxacin Ophthalmic prescriptions shown $15,307 gross reimbursement (before rebates) ≈ $39 per prescription (gross)

    Summed across the 1 of 10 listed NDC products with Medicaid activity — every brand and generic of this exact strength & form. RxNorm 992395

    Shares are of the Medicaid prescriptions shown here. Product grouping follows RxNorm (the National Library of Medicine’s drug terminology), so “one product” means one strength & dosage form regardless of manufacturer. Dollar figures are gross Medicaid reimbursement before mandatory rebates — rebates (often large, especially for brand-name drugs) are confidential, so actual net cost to Medicaid is lower than shown.

    Source: Medicaid State Drug Utilization Data (CMS), aggregated by generic ingredient — summed across every NDC (all brands, strengths, salt forms and dosage forms) of Gatifloxacin Ophthalmic, and across all states and both fee-for-service and managed-care claims. A general popularity signal; it excludes Medicare, commercial insurance and cash prescriptions, so it is not total U.S. use. Based on the 1 of 10 listed Gatifloxacin Ophthalmic NDCs with Medicaid activity.

    🔍 Compare Gatifloxacin Ophthalmic products

    A representative set of FDA-listed product records for Gatifloxacin Ophthalmic — across manufacturers, strengths, and dosage forms, grouped by form with each product’s manufacturer and how the FDA approved it. The same medicine may be made and packaged by different companies, so a single drug can have many directory entries. (It’s also why a refill can look different — a new shape, color, or box — even though it contains the same medication.)

    Strength Route Manufacturer / Labeler Category ⓘ Details
    💊Eye drops
    5 mg/mL Ophthalmic Akorn ANDA View NDC →
    5 mg/mL Ophthalmic Allergan, Inc. × 3 listings NDA View NDC →
    5 mg/mL Ophthalmic Caplin Steriles Limited ANDA View NDC →
    5 mg/mL Ophthalmic Leading Pharma, LLC ANDA View NDC →
    5 mg/mL Ophthalmic Lupin Pharmaceuticals, Inc. ANDA View NDC →
    5 mg/mL Ophthalmic Pacific Pharma, Inc. × 2 listings NDA AUTHORIZED GENERIC View NDC →
    5 mg/mL Ophthalmic Sandoz Inc × 2 listings ANDA View NDC →
    5 mg/mL Ophthalmic Torrent Pharmaceuticals Limited ANDA View NDC →

    Showing 12 of 12 products — FDA National Drug Code Directory. See every product, package size and price: browse all 12 Gatifloxacin Ophthalmic NDCs →

    RxNorm Concept Web — From Ingredient to Every Form and Strength

    This page starts with one ingredient concept (IN). The branches below show its dose-form concepts (SCDF), then the available clinical drug and strength concepts (SCD). Combination products remain separate concepts with their own pages.

    Ingredient (IN) Gatifloxacin Ophthalmic RxCUI 228476 3 dose forms · 5 strengths
    1. Dose form (SCDF) Ophthalmic Solution RxCUI 402433 In current FDA listings
      Clinical drug / strength (SCD) 3 MG/ML RxCUI 402089 5 MG/ML RxCUI 992395
    2. Dose form (SCDF) Oral Suspension RxCUI 644540 No current FDA listing
      Clinical drug / strength (SCD) 40 MG/ML RxCUI 644541
    3. Dose form (SCDF) Oral Tablet RxCUI 374621 No current FDA listing
      Clinical drug / strength (SCD) 200 MG RxCUI 310445 400 MG RxCUI 314009

    Look up RxCUI 228476 in the RxCUI Atlas →

    RxNorm is the U.S. National Library of Medicine’s normalized drug vocabulary. Its concept hierarchy can include forms that are not currently marketed; the status on each branch compares that concept with current FDA listings. RxCUIs identify vocabulary concepts, not individual packages or manufacturers.

    🏷️ Sold under these brand names

    Zymaxid Zymar

    🏭 Manufacturers & labelers

    Allergan, Inc. 3 Pacific Pharma, Inc. 2 Sandoz Inc 2 Akorn 1 Caplin Steriles Limited 1 Leading Pharma, LLC 1 Lupin Pharmaceuticals, Inc. 1 Torrent Pharmaceuticals Limited 1

    RxNorm drug class

    Gatifloxacin Ophthalmic belongs to the Quinolone Antimicrobial class.

    Pharmacologic class Quinolone Antimicrobial
    Drug family (ATC) Fluoroquinolones, Fluoroquinolones

    Classified by RxNorm RxClass — the U.S. National Library of Medicine's standardized drug-classification service (Established Pharmacologic Class from the FDA, the ATC drug family from the WHO, and mechanism of action). Reference only, not medical advice.

    🔬 Where this comes from

    Core label, product, RxNorm, safety, and utilization data on this page come from the sources identified below. AI-written, editorial, and licensed sections are labeled separately.

    📄
    FDA-filed drug labels (SPL) Uses, dosing, warnings & side effects from SPL records retrieved through openFDA; the linked representative set can be verified on DailyMed. ✓ Linked label effective Sep 8, 2016
    🏭
    Forms, brands & labelersAggregated from ingredient-matched FDA National Drug Code Directory product records for Gatifloxacin Ophthalmic.
    📈
    Real-world reportsThe FDA Adverse Event Reporting System (FAERS), served through openFDA.
    🚨
    Recalls & shortagesopenFDA drug-enforcement reports and the FDA drug-shortage database.
    🧾 Clinical label set — FDA-filed SPL labels retained for Gatifloxacin Ophthalmic after exact ingredient or ingredient-combination matching and applicable route/form matching
    Clinical labels in scope
    5
    NDC products indexed
    12
    Distinct labelers/manufacturers represented
    8
    Linked representative label ⓘ
    Allergan, Inc.
    Linked label effective
    Sep 8, 2016
    Composite sections available
    19
    Linked SPL Set ID
    1160b16c-929a-4e85-9c0b-1d8c96a7678b
    Linked SPL Document ID
    96056904-df3f-43e9-a3bd-8bb7d19eb49c
    Open the linked representative label on DailyMed ↗

    How we combine label and product data

    HelloPharmacist combines public FDA and NLM records; we don’t author the underlying clinical facts. We identified 5 FDA-filed SPL label sets within the page’s selected clinical scope after exact ingredient or ingredient-combination matching and applicable route/form matching. The representative label is the starting point for the displayed reference monograph; the 12 largest stored in-scope SPL records, which may include that representative, are compared section by section, and the longest available version of each section is retained. Forms, routes, brands, labelers, product-listed strengths, and product-record counts are aggregated separately from ingredient-matched FDA NDC Directory records; package records listed above are associated with the linked SPL; and the normalized concept hierarchy comes from NLM RxNorm.

    Where a section is identified as AI-written, its plain-language text is generated from bounded label evidence. New draft drug pages remain in the admin review queue before first publication. Allergan, Inc. is the representative DailyMed label linked for verification and dates; it is not the sole source used for the page.

    This is general education, not medical advice — always consult your doctor or pharmacist about your medications and any medical condition. For the exact wording of the linked representative label, view that label on DailyMed; some displayed composite sections may come from other in-scope SPL labels. Learn how we use AI and our data sources & update cadence.