HomeNDC LookupIngredientsNorethindrone Acetate › 68462-0304-50
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Norethindrone Acetate 5 mg Tablet, 50-count

by Glenmark Pharmaceuticals Inc., USA · 50 TABLET in 1 BOTTLE (68462-304-50)
NDC 68462-0304-50
🏷️ FDA NDC (as labeled) 68462-304-50 billing pads the product segment with a zero
This package
Contains50-count Cost per ea$0.2948 NADAC Per package$14.74 / 50 tablets Pack sizes2 compare ↓
Also priced by: Medicaid pays $0.4714/unit · Part D plans $0.4972/unit — full pricing hub ↓
Also comes in: 500 tablets 68462-0304-05
Rx only Generic On market Non-controlled
🗂️ Data synced Jul 24, 2026 · sources: openFDA · FDA label (DailyMed) · FDA Orange & Purple Book · First Databank · CMS NADAC, ASP, Medicare & Medicaid · RxNorm
📋 All sources & update times →

🆔 Identity & classification

FDA NDC (as labeled) 68462-304-50
Product NDC 68462-304
11-digit billing NDC 68462030450
NCPDP billing unit EA — each (per item)
RxCUI 1000405
UNII 9S44LIC7OJ
UPC 0368462304501
Application # ANDA091090
SPL Set ID d0a94321-eb60-4aa6-a429-f0156f9f8e01
Established class (EPC) Progestin
Chemical class Progesterone Congeners
DEA schedule Non-controlled
Marketing category ANDA
Marketing status On market
FDA listing status Listed (active directory)
Marketing start 2010-07-21
Route ORAL
Dosage form TABLET
Substance NORETHINDRONE ACETATE
GPI-14 26000030100305
GPI class Norethindrone Acetate
GCN Seq No 003274
GCN 11280
HICL code 001443
Ingredient (HICL) Norethindrone Acetate
HIC1 code G
Therapeutic class — broad (HIC1) Female Genital System
HIC2 code G2
Therapeutic class — intermediate (HIC2) Progestogens
HIC3 code G2A
Therapeutic class — specific (HIC3) Progestational Agents
AHFS code 68:32.00.00
AHFS class Progestins
FDB label name NORETHINDRONE 5 MG TABLET
FDB brand name Norethindrone Acetate
Legend status F — Federal legend — prescription drug or device
TE code (Orange Book) AB · RLD · RS
Why two NDCs? The FDA registers this code as 68462-304-50 — a 5-3-2 layout, and that's what's printed on the package and shown on DailyMed. For insurance claims, every NDC is standardized to a uniform 11-digit 5-4-2 format by adding a zero to the product segment → 68462-0304-50. Same drug, same package — only the format differs.
Where does this data come from?
Identifiers from the FDA openFDA NDC Directory and Structured Product Labeling; RxCUI from RxNorm (NLM); GPI from Medi-Span; GCN / HIC / AHFS / legend from First Databank.

🏷️ RxNorm drug class

This medicine belongs to the Progestin class.

Pharmacologic class Progestin
Drug family (ATC) Progestogens and estrogens, sequential preparations, Progestogens, Estren derivatives
Where does this data come from?
Therapeutic classes from RxNorm RxClass (U.S. National Library of Medicine) — Established Pharmacologic Class (FDA), ATC drug family (WHO) and mechanism of action, matched by this product’s RxCUI.

🏭 Manufacturer & labeler

LabelerGlenmark Pharmaceuticals Inc., USA
Application holderGLENMARK PHARMACEUTICALS LTD
FDA applicationANDA091090 (ANDA)
Labeler code68462
First marketedJul 2010
Product typeHuman Prescription Drug
Portfolio343 products on file
The labeler markets the product; the application holder owns the FDA approval. They’re often the same company but can differ (e.g. a repackager or an authorized generic). A mailing address / phone appears here when the manufacturer includes it in the product’s FDA label (not all do).
Where does this data come from?
Labeler, application holder and registered establishment from the FDA openFDA NDC Directory and Drugs@FDA; address/contact from the product’s FDA label.

🩺 Clinical

Label name NORETHINDRONE 5 MG TABLET Ingredient Norethindrone Acetate
📗 Our plain-language guide HelloPharmacist
  • It depends on the product. Most norethindrone tablets — including brands like Camila, Errin, Emzahh, and Affodel — are progestin-only birth control pills taken daily to prevent pre...
  • Regular combination birth control pills contain two hormones — estrogen and progestin. Norethindrone is a progestin-only pill, sometimes called the 'mini-pill.' Because it has no e...
  • How is this different from regular birth control pills?
  • The most common thing people notice is irregular bleeding — spotting between periods, or changes in your cycle. Headache, breast tenderness, nausea, and dizziness are also reported...
📖 Read our full Norethindrone guide →
Where does this data come from?
Plain-language summary from MedlinePlus (U.S. National Library of Medicine); supplement & herbal interactions and nutrient depletion data from the Natural Medicines database; our full guide is HelloPharmacist editorial content.

💊 What it looks like

Color White
ShapeOval
ImprintG;304
Size11 mm
ScoringScored — splits in 2
One label can cover several strengths, so colors may be combined — always confirm a loose pill against the dispensed prescription label or a pharmacist.
Where does this data come from?
Physical description (imprint, shape, color, scoring, coating) from this product’s FDA Structured Product Labeling (SPL), mirrored from DailyMed / openFDA.

🧪 Inactive Ingredients / Excipients

Inactive ingredients, also called excipients, are components of the drug product other than the active ingredient. They may include fillers, dyes, coatings, preservatives, flavors, or other formulation ingredients.

💡 Tap an ingredient (hover on desktop) to see what it is and why it’s used.

  • UNII EWQ57Q8I5X
    Lactose monohydrate is a natural sugar derived from milk. It serves as a filler and binder in tablets and capsules, helping create the proper size, texture, and consistency of the medicine.
  • UNII 70097M6I30
    Magnesium stearate is a salt made from magnesium and stearic acid, a fatty substance. It's used in tablets and capsules as a lubricant and glidant to help ingredients flow smoothly during manufacturing and prevent sticking.
  • UNII OP1R32D61U
    Microcrystalline cellulose is a purified form of cellulose, a natural fiber from plant sources. It acts as a binder and filler in tablets and capsules, helping hold ingredients together and give the medicine its shape and size.
  • UNII ETJ7Z6XBU4
    Silicon dioxide is a naturally occurring mineral used as a glidant and anti-caking agent. It helps powder ingredients flow smoothly and prevents clumping during manufacturing and storage.
  • UNII 7SEV7J4R1U
    A powder made from a naturally occurring mineral. In medicines, talc works as a glidant and anti-caking agent, helping tablets and capsules flow smoothly during manufacturing and preventing clumping.

5 inactive ingredients listed in the exact product block matched to this NDC.

Where does this data come from?
Data sourced from official FDA Structured Product Labeling (SPL) via DailyMedingredient classCode="IACT" elements from the exact product block matched by this NDC. Label-section narrative from DailyMed / the openFDA label index is shown separately when available.

Inactive ingredient FAQ

Are inactive ingredients the same for every manufacturer?
No. Inactive ingredients can differ by manufacturer, dosage form, strength, and package / product version.
Why might an inactive ingredient be missing?
Some SPLs do not provide a complete structured inactive-ingredient list, and older or unusual labels may only include the information in narrative text.
Can inactive ingredients matter?
Yes. They can matter for allergies, intolerances, dyes, gluten / lactose concerns, preservatives, and formulation differences — but confirm with a pharmacist or the manufacturer when it’s clinically important.

💲 Pricing

A drug doesn't have one price. Each row is a different public payment system, and none is what you'd pay at the counter — that depends on your insurance. The ⓘ on each row explains what it measures.

Price systemPer eaPer package
Retail pharmacies payNADAC · weekly $0.295 $14.74 / 50 tablets
Medicaid paysCMS SDUD · 12 mo $0.4714 $23.57 / 50 tablets
Medicare drug plans payPart D · Q2 2026 $0.4972 $24.86 / 50 tablets
NADAC price history (per ea) — tap or hover for the price & month
Dec 2021 Jul 2022 Dec 2025 Aug 2026 $0.600 $0.290
▼ Down 48% over the last 24 months.
Where does this data come from?
NADAC (National Average Drug Acquisition Cost) is the CMS weekly pharmacy-acquisition-cost survey — what pharmacies pay. ASP (Average Sales Price) is the CMS Medicare Part B drug-payment file, published quarterly. Medicaid pays is computed by us from CMS State Drug Utilization Data (total reimbursed ÷ units, trailing 12 months) — gross of rebates and inclusive of dispensing fees, so it reflects what Medicaid paid, not an acquisition cost. Medicare drug plans pay is the median negotiated point-of-sale unit cost across plans listing this NDC in the CMS quarterly Prescription Drug Plan pricing files, before rebates. The VA pays is the federal contract price (FSS, and the statutory Big 4 ceiling where listed) from the VA National Acquisition Center pharmaceutical price file. All are free public government data; each measures a different payer, so the figures are not directly comparable.

🔁 Therapeutic equivalents

ProductLabelerPackNADAC/unitTEStatusPrice vs. this
Norethindrone Acetate 5 mg 00555-0211-10 Teva 50 tablets $0.295 AB Availability likely
Norethindrone acetate 5 mg 50742-0267-50 Ingenus 50 tablets $0.295 AB Availability likely
Norethindrone Acetate 5 mg 60687-0921-21 American 30 tablets $0.295 AB Availability likely
Norethindrone Acetate 5 mgthis 68462-0304-50 Glenmark 50 tablets $0.295 AB Availability likely
Gallifrey 5 mg 70700-0326-50 Xiromed 50 tablets $0.295 AB Availability likely
Norethindrone Acetate 5 mg 42291-0650-90 AvKARE 90 tablets AB FDA listed
Norethindrone Acetate 5 mg 51407-0599-50 Golden 50 tablets AB FDA listed
Norethindrone Acetate 5 mg 65162-0475-03 Amneal 30 tablets AB FDA listed
About this product: this is a generic version of the medicine. FDA equivalence ratings are shown when available, and other versions are listed above, least expensive first.
Where does this data come from?
Equivalents are other NDCs of the same ingredient, form and route from the openFDA NDC Directory, ranked least-expensive-first by NADAC. Therapeutic-equivalence (AB) ratings come from the FDA Orange Book; biologics use the FDA Purple Book for biosimilar & interchangeable status.

Availability & generic status

🏛️
2010
On the market since
Jul 2010
📍
2026
Currently FDA-listed
16 years listed
🔓
·
Generic on the market
this product is a generic
This is a generic drug

This product is an FDA-approved generic. Other versions of the same drug are listed under Therapeutic equivalents, least expensive first.

Where does this data come from?
Patents and exclusivity from the FDA Orange Book (small-molecule drugs), refreshed from public FDA data. Generic launch timing is an estimate, not a guarantee.

🗺️ Medicaid utilization & spend

📍 This exact package only: Medicaid data is reported per full 11-digit NDC — labeler, product and pack size — so every number here is for 68462-0304-50, not the drug overall. Other pack sizes report separately.
💊 Pharmacy benefit only: These are Medicaid outpatient pharmacy claims, billed by NDC. They exclude the medical benefit — clinic- or hospital-administered drugs billed under HCPCS J-codes — so drugs used mostly that way (e.g. Avastin, Lucentis, Keytruda) can look low or missing here. That’s expected, not an error.
📅 Q1 2025 – Q4 2025 · 4 quarters of data
ⓘ The newest quarter is usually incomplete when first published; states restate recent quarters in later CMS releases, so the latest figures typically revise upward. State coverage-policy changes can also shift quarter-to-quarter totals.
Prescriptions last 4 qtrs
158.6K
Units reimbursed last 4 qtrs
8M
Gross reimbursed last 4 qtrs
$3.77M
Avg / prescription
$23.81
Avg / unit
$0.4714
Latest quarter Q4 2025
38.9KRx
Medicaid pays / ea
$0.4714
gross reimbursed
vs
NADAC / ea
$0.2948
acquisition cost
=
Spread
+$0.1766
+60% vs cost
What Medicaid paid per ea (before rebates; includes the pharmacy’s dispensing fee) compared with NADAC — the average price pharmacies pay to buy the drug. A positive spread means Medicaid reimbursed more than the purchase price, before manufacturer rebates.
Fee-for-service vs managed care
35% FFS 65% MCO
Fee-for-service · 54,870 Rx Managed care · 103,686 Rx
State Medicaid map
Alaska: 14,565 units · 1,987 per 100k residents AK Maine: 104,153 units · 7,466 per 100k residents ME Washington: 345,150 units · 4,418 per 100k residents WA Idaho: 18,814 units · 958 per 100k residents ID Montana: 46,980 units · 4,150 per 100k residents MT North Dakota: 7,796 units · 996 per 100k residents ND Minnesota: 117,507 units · 2,048 per 100k residents MN Wisconsin: 127,492 units · 2,157 per 100k residents WI Michigan: 385,087 units · 3,837 per 100k residents MI New York: 882,266 units · 4,508 per 100k residents NY Vermont: 45,942 units · 7,101 per 100k residents VT New Hampshire: 66,051 units · 4,711 per 100k residents NH Oregon: 217,275 units · 5,133 per 100k residents OR Nevada: 33,405 units · 1,046 per 100k residents NV Wyoming: 6,323 units · 1,083 per 100k residents WY South Dakota: 20,636 units · 2,245 per 100k residents SD Iowa: 144,425 units · 4,503 per 100k residents IA Illinois: 29,872 units · 238 per 100k residents IL Indiana: 168,024 units · 2,449 per 100k residents IN Ohio: 458,747 units · 3,893 per 100k residents OH Pennsylvania: 465,338 units · 3,590 per 100k residents PA New Jersey: 141,229 units · 1,520 per 100k residents NJ Massachusetts: 548,568 units · 7,836 per 100k residents MA California: 170,776 units · 438 per 100k residents CA Utah: 118,788 units · 3,476 per 100k residents UT Colorado: 261,995 units · 4,457 per 100k residents CO Nebraska: 26,098 units · 1,319 per 100k residents NE Missouri: 136,580 units · 2,204 per 100k residents MO Kentucky: 217,814 units · 4,813 per 100k residents KY West Virginia: 81,340 units · 4,595 per 100k residents WV Virginia: 325,836 units · 3,738 per 100k residents VA Maryland: 134,778 units · 2,181 per 100k residents MD Connecticut: 237,148 units · 6,556 per 100k residents CT Rhode Island: 61,362 units · 5,604 per 100k residents RI Arizona: 152,987 units · 2,059 per 100k residents AZ New Mexico: 58,893 units · 2,786 per 100k residents NM Kansas: 29,523 units · 1,004 per 100k residents KS Arkansas: 116,335 units · 3,793 per 100k residents AR Tennessee: 20,491 units · 288 per 100k residents TN North Carolina: 479,942 units · 4,430 per 100k residents NC South Carolina: 129,236 units · 2,405 per 100k residents SC Delaware: 26,829 units · 2,602 per 100k residents DE Oklahoma: 100,537 units · 2,481 per 100k residents OK Louisiana: 45,550 units · 996 per 100k residents LA Mississippi: 34,511 units · 1,174 per 100k residents MS Alabama: 89,220 units · 1,747 per 100k residents AL Georgia: 269,415 units · 2,443 per 100k residents GA D.C.: 40,897 units · 6,023 per 100k residents DC Hawaii: 1,314 units · 91.6 per 100k residents HI Texas: 137,390 units · 450 per 100k residents TX Florida: 104,779 units · 463 per 100k residents FL
Units reimbursed · per 100k residents
91.67,836
gray = no data reported
Colors are per 100,000 residents, so big states don’t automatically dominate. Tap or hover a state for its actual totals.
Tap or hover a state
…for its Medicaid breakdown
🏆 Top states by units · per 100k residents
1 Massachusetts 7,836 /100k
2 Maine 7,466 /100k
3 Vermont 7,101 /100k
4 Connecticut 6,556 /100k
5 D.C. 6,023 /100k
6 Rhode Island 5,604 /100k
7 Oregon 5,133 /100k
8 Kentucky 4,813 /100k
National units — by quarter
💵 About the dollar figures: “reimbursed” is what Medicaid paid pharmacies before confidential manufacturer rebates, so the program’s real net cost is lower than these numbers. Fee-for-service and managed-care claims are combined unless split above. Source: CMS State Drug Utilization Data; per-100k rates use 2023 Census population estimates.

💊 Medicaid utilization by pack size

Medicaid (SDUD) totals over the four most recent reported quarters for every package size of this drug — handy when a specific package (e.g. a starter/titration pack) carries little or no Medicaid volume on its own.
50 tablets this page68462-0304-50 158,556 Rx · $3,774,772
500 tablets68462-0304-05 No Medicaid data
Drug total (last 4 qtrs): 158,556 Rx · 8,007,371 units · $3,774,772 gross reimbursed
Tap a pack size to open its page. Source: CMS State Drug Utilization Data, last 4 quarters.

📊 Medicare Part D spend CMS · PART D · 2026 (Q1)

Medicare Part D (outpatient prescription) spending for Norethindrone Acetate — the program that covers self-administered drugs. 4 manufacturers.
⚠️ Drug-level data: CMS publishes Part D spending by drug, not by NDC — these figures combine every manufacturer, strength and package size sold under the name Norethindrone Acetate. That’s a different level of aggregation than the Medicaid card above, which is specific to this exact 11-digit NDC (pack size included), so the two aren’t directly comparable.
Period
Total Part D spend
$565.1K
Claims incl. refills
14.2K
Beneficiaries
8.9K
Spend / beneficiary
$63.32
Spend / claim
$39.71
Trend by period
💵 About the dollar figures: spending is what Part D plans paid before confidential manufacturer rebates, so the program’s real net cost is lower. A blank patient count means fewer than 11 people — CMS hides counts that small to protect privacy. Source: CMS Medicare Quarterly Part D Spending by Drug (data.cms.gov), updated quarterly.

📦 Packaging — all sizes for this product

Package NDCDescription Per unit Per pack Marketing startStatus
68462-0304-05 500 TABLET in 1 BOTTLE (68462-304-05) 2010-07-21 Active
68462-0304-50 You're viewing this 50 TABLET in 1 BOTTLE (68462-304-50) $0.2948 / ea $14.74 2010-07-21 Active

You're viewing the smallest of 2 pack sizes for this product.

In Medicaid, this is the most-dispensed pack of this product — about 100% of fills over the last four reported quarters. See all packs ↓

Pack size FAQ

What quantity is in NDC 68462-0304-50?
NDC 68462-0304-50 is a 50-count package — 50 tablet in 1 bottle.
What is the difference between NDC 68462-0304-50 and NDC 68462-0304-05?
Both are Norethindrone Acetate 5 mg Tablet — the drug itself is identical. NDC 68462-0304-50 is the 50-count package, while NDC 68462-0304-05 is the 500 tablets package.
What NDC number is used to bill for this package of Norethindrone Acetate 5 mg Tablet?
Bill NDC 68462-0304-50 — the 11-digit billing format is 68462030450. Pharmacy and medical claims use the 11-digit form; the FDA label may print a shorter form of the same code.

Prices are the latest CMS NADAC pharmacy acquisition cost per NDC; per-pack figures are per-unit × pack quantity, shown only when the pack is denominated in the same measure NADAC prices.

📄 Full prescribing information FDA SPL

The complete FDA label for this product — the official prescribing information, verbatim, section by section. Jump with a chip, search within the label, or expand everything.
🎯 Indications and Usage 56 words

INDICATIONS AND USAGE Norethindrone acetate is indicated for the treatment of secondary amenorrhea, endometriosis, and abnormal uterine bleeding due to hormonal imbalance in the absence of organic pathology, such as submucous fibroids or uterine cancer. Norethindrone acetate is not intended, recommended or approved to be used with concomitant estrogen therapy in postmenopausal women for endometrial protection.

⏱️ Dosage and Administration 159 words

DOSAGE AND ADMINISTRATION Therapy with norethindrone acetate must be adapted to the specific indications and therapeutic response of the individual patient. Secondary amenorrhea, abnormal uterine bleeding due to hormonal imbalance in the absence of organic pathology: 2.5 to 10 mg norethindrone acetate may be given daily for 5 to 10 days to produce secretory transformation of an endometrium that has been adequately primed with either endogenous or exogenous estrogen. Progestin withdrawal bleeding usually occurs within three to seven days after discontinuing norethindrone acetate therapy.

Patients with a past history of recurrent episodes of abnormal uterine bleeding may benefit from planned menstrual cycling with norethindrone acetate. Endometriosis: Initial daily dosage of 5 mg norethindrone acetate for two weeks. Dosage should be increased by 2.5 mg per day every two weeks until 15 mg per day of norethindrone acetate is reached.

Therapy may be held at this level for six to nine months or until annoying breakthrough bleeding demands temporary termination.

Contraindications 82 words

CONTRAINDICATIONS • Known or suspected pregnancy. There is no indication for norethindrone acetate in pregnancy. (See PRECAUTIONS ). • Undiagnosed vaginal bleeding • Known, suspected or history of cancer of the breast • Active deep vein thrombosis, pulmonary embolism or history of these conditions • Active or recent (e.g., within the past year) arterial thromboembolic disease (e.g., stroke, myocardial infarction) • Impaired liver function or liver disease • As a diagnostic test for pregnancy • Hypersensitivity to any of the drug components

⚠️ Warnings 82 words

WARNINGS 1. Cardiovascular disorders Patients with risk factors for arterial vascular disease (e.g., hypertension, diabetes mellitus, tobacco use, hypercholesterolemia, and obesity) and/or venous thromboembolism (e.g., personal history or family history of VTE, obesity, and systemic lupus erythematosus) should be managed appropriately. 2.

Visual abnormalities Discontinue medication pending examination if there is a sudden partial or complete loss of vision or if there is sudden onset of proptosis, diplopia, or migraine. If examination reveals papilledema or retinal vascular lesions, medication should be discontinued.

🤒 Adverse Reactions 132 words

ADVERSE REACTIONS See WARNINGS and PRECAUTIONS . The following adverse reactions have been observed in women taking progestins: • Breakthrough bleeding • Spotting • Change in menstrual flow • Amenorrhea • Edema • Changes in weight (decreases, increases) • Changes in the cervical squamo-columnar junction and cervical secretions • Cholestatic jaundice • Rash (allergic) with and without pruritus • Melasma or chloasma • Clinical depression • Acne • Breast enlargement/tenderness • Headache/migraine • Urticaria • Abnormalities of liver tests (i.e., AST, ALT, Bilirubin) • Decreased HDL cholesterol and increased LDL/HDL ratio • Mood swings • Nausea • Insomnia • Anaphylactic/anaphylactoid reactions • Thrombotic and thromboembolic events (e.g., deep vein thrombosis, pulmonary embolism, retinal vascular thrombosis, cerebral thrombosis and embolism) • Optic neuritis (which may lead to partial or complete loss of vision)

🔄 Drug / Laboratory Test Interactions 217 words

3. Drug/Laboratory Tests Interactions The following laboratory test results may be altered by the use of estrogen/progestin combination drugs: • Accelerated prothrombin time, partial thromboplastin time, and platelet aggregation time; increased platelet count; increased factors II, VII antigen, VIII antigen, VIII coagulant activity, IX, X, XII, VII-X complex, II-VII-X complex, and beta-thromboglobulin; decreased levels of antifactor X a and antithrombin III, decreased antithrombin III activity; increased levels of fibrinogen and fibrinogen activity; increased plasminogen antigen and activity. • Increased thyroid-binding globulin (TBG) levels leading to increased circulating total thyroid hormone levels as measured by protein-bound iodine (PBI), T 4 levels (by column or by radioimmunoassay) or T 3 levels by radio immunoassay.

T 3 resin uptake is decreased, reflecting the elevated TBG. Free T 4 and free T 3 concentrations are unaltered. Patients on thyroid replacement therapy may require higher doses of thyroid hormone. • Other binding proteins may be elevated in serum (i.e., corticosteroid binding globulin (CBG), sex hormone binding globulin (SHBG)) leading to increased circulating corticosteroid and sex steroids, respectively.

Free or biologically active hormone concentrations are unchanged. Other plasma proteins may be increased (angiotensinogen/renin substrate, alpha-1-antitrypsin, ceruloplasmin). • Increased plasma HDL and HDL 2 cholesterol subfraction concentrations, reduced LDL cholesterol concentration, increased triglycerides levels. • Impaired glucose metabolism. • Reduced response to metyrapone test.

🤰 Pregnancy 59 words

5. Pregnancy Category X Norethindrone acetate is contraindicated during pregnancy as it may cause fetal harm when administered to pregnant women. Several reports suggest an association between intrauterine exposure to progestational drugs in the first trimester of pregnancy and congenital abnormalities in male and female fetuses. Some progestational drugs induce mild virilization of the external genitalia of female fetuses.

🧒 Pediatric Use 11 words

7. Pediatric Use Norethindrone acetate tablets are not indicated in children.

🧬 Clinical Pharmacology ~2 min read

CLINICAL PHARMACOLOGY Norethindrone acetate induces secretory changes in an estrogen-primed endometrium. On a weight basis, it is twice as potent as norethindrone. PHARMACOKINETICS Absorption: Norethindrone acetate is completely and rapidly deacetylated to norethindrone (NET) after oral administration, and the disposition of norethindrone acetate is indistinguishable from that of orally administered norethindrone.

Norethindrone acetate is rapidly absorbed from norethindrone acetate tablets, with maximum plasma concentration of norethindrone generally occurring at about 2 hours post-dose. The pharmacokinetic parameters of norethindrone following single oral administration of norethindrone acetate in 29 healthy female volunteers are summarized in Table 1. Table 1 Pharmacokinetic Parameters after a Single Dose of Norethindrone Acetate in Healthy Women Norethindrone Acetate (n=29) Arithmetic Mean ± SD Norethindrone (NET) AUC (0-inf) (ng/ml*h) 166.90 ±

56.28C max (ng/ml) 26.19 ± 6.19 t max (h) 1.83 ± 0.58 t 1/2 (h) 8.51 ±

2.19AUC = area under the curve, C max = maximum plasma concentration, t max = time at maximum plasma concentration, t 1/2 = half-life, SD = standard deviation Figure 1. Mean Plasma Concentration Profile after a Single Dose of 5 mg Administered to 29 Healthy Female Volunteers under Fasting Conditions figure1 Effect of Food: The effect of food administration on the pharmacokinetics of norethindrone acetate has not been studied. Distribution: Norethindrone is 36% bound to sex hormone-binding globulin (SHBG) and 61% bound to albumin.

Volume of distribution of norethindrone is about 4 L/kg. Metabolism: Norethindrone undergoes extensive biotransformation, primarily via reduction, followed by sulfate and glucuronide conjugation. The majority of metabolites in the circulation are sulfates, with glucuronides accounting for most of the urinary metabolites.

Excretion: Plasma clearance value for norethindrone is approximately

0.4L/hr/kg. Norethindrone is excreted in both urine and feces, primarily as metabolites. The mean terminal elimination half-life of norethindrone following a single dose administration of norethindrone acetate is approximately 9 hours.

SPECIAL POPULATIONS Geriatrics The effect of age on the pharmacokinetics of norethindrone after norethindrone acetate administration has not been evaluated. Race The effect of race on the disposition of norethindrone after norethindrone acetate administration has not been evaluated. Renal Insufficiency The effect of renal disease on the disposition of norethindrone after norethindrone acetate administration has not been evaluated.

In pre-menopausal women with chronic renal failure undergoing peritoneal dialysis who received multiple doses of an oral contraceptive containing ethinyl estradiol and norethindrone, plasma norethindrone concentration was unchanged compared to concentrations in pre-menopausal women with normal renal function. Hepatic Insufficiency The effect of hepatic disease on the disposition of norethindrone after norethindrone acetate administration has not been evaluated. However, norethindrone acetate is contraindicated in markedly impaired liver function or liver disease.

Drug Interactions No pharmacokinetic drug interaction studies investigating any drug-drug interactions with norethindrone acetate have been conducted.

📦 How Supplied / Storage and Handling 47 words

HOW SUPPLIED Norethindrone acetate tablets USP are available as: 5 mg: White to off-white oval, flat faced beveled edged, uncoated tablets debossed with ‘G with breakline’ on one side and 304 on other side. Available as follows: Bottles of 50 NDC 68462-304-50 Bottles of 500 NDC 68462-304-05

📦 Storage and Handling 30 words

Store at 20° to 25°C (68° to 77°F) [See USP Controlled Room Temperature]. Distributed by: Glenmark Pharmaceuticals Inc., USA Elmwood Park, NJ 07407 Questions? 1 (888)721-7115 www.glenmarkpharma-us.com August 2025 glenmarklogo1

📋 Description 59 words

DESCRIPTION Norethindrone acetate tablets USP - 5 mg oral tablets. Norethindrone acetate USP, (17-hydroxy-19-nor-17α-pregn-4-en-20-yn-3-one acetate), a synthetic, orally active progestin, is the acetic acid ester of norethindrone. It is a white, or creamy white, crystalline powder.

Norethindrone acetate tablets USP, 5 mg contain the following inactive ingredients: colloidal silicon dioxide, lactose monohydrate, magnesium stearate, microcrystalline cellulose and talc. structure

💬 Information for Patients 23 words

2. Information for the Patient Healthcare providers are advised to discuss the PATIENT INFORMATION leaflet with patients for whom they prescribe norethindrone acetate.

Source: FDA Structured Product Labeling, mirrored from DailyMed / openFDA. Prefer the government’s original formatting? View this label on DailyMed ↗
For educational and professional reference only — not medical advice. Pricing reflects published NADAC and CMS ASP (free public data) and may differ from your acquisition cost; always verify before billing or dispensing.