Teriflunomide
31 interactions 1 explained in plain EnglishTeriflunomide is used to treat adults with various forms of multiple sclerosis (MS; a disease in which the nerves do not function properly and people may experience weakness, numbness, loss of muscle coordination, and problems with vision, speech, and bladder control) including: clinically isolated syndrome (CIS; nerve… Read the full Teriflunomide drug information page →
Sources: FDA prescribing information (Structured Product Labeling), the published literature cited in each entry, DDInter 2.0 (a major open-access drug-interaction database), and legacy DrugBank interaction data distributed by the NIH's RxNav service (decommissioned in 2024) — analyzed and reviewed by our pharmacist team. How we build this library →
Major
Teriflunomide Simvastatin Flolipid Explained Increased exposure of OATP1B1/1B3 substrate Details Teriflunomide Acyclovir Avaclyr Increased exposure of OAT3 substrate Details Teriflunomide Acyclovir Injection Avaclyr Increased exposure of OAT3 substrate Details Teriflunomide Acyclovir Ophthalmic Avaclyr Increased exposure of OAT3 substrate Details Teriflunomide Acyclovir Topical Zovirax Increased exposure of OAT3 substrate Details Teriflunomide Alpelisib Piqray Increased alpelisib exposure and an increased risk of alpelisib-related adverse effects and toxicity Details Teriflunomide Asciminib Scemblix Increased BCRP substrate exposure and an increased risk of BCRP substrate-related adverse effects Details Teriflunomide Aztreonam Injection Azactam Increased risk of aztreonam exposure Details Teriflunomide Atorvastatin Atorvaliq Increased exposure of OATP1B1/1B3 substrate Details Teriflunomide Baricitinib Olumiant Increased exposure of OAT3 substrate Details Teriflunomide Cefaclor Ceclor® Increased exposure of OAT3 substrate Details Teriflunomide Daprodustat Jesduvroq Increased daprodustat exposure Details Teriflunomide Finerenone Kerendia Increased finerenone exposure and an increased risk of finerenone-related adverse effects Details Teriflunomide Furosemide Injection Disal Increased exposure of OAT3 substrate Details Teriflunomide Irinotecan Camptosar Increased exposure of BCRP substrate Details Teriflunomide Irinotecan Injection Camptosar Increased exposure of BCRP substrate Details Teriflunomide Leniolisib Joenja Increased BCRP substrate exposure Details Teriflunomide Letermovir Injection Prevymis Increased exposure of OATP1B1/1B3 substrate Details Teriflunomide Loperamide Diamode Increased loperamide exposure and an increased risk of loperamide-related adverse effects Details Teriflunomide Methotrexate Jylamvo Increased exposure of methotrexate and increased risk of hepatotoxicity and bone marrow toxicity Details Teriflunomide Methotrexate Injection Abitrexate® Increased exposure of methotrexate and increased risk of hepatotoxicity and bone marrow toxicity Details Teriflunomide Methylergonovine Methergine Increased methylergonovine exposure Details Teriflunomide Montelukast Singulair Increased exposure of CYP2C8 substrate Details Teriflunomide Nifedipine Adalat® Increased NIFEdipine exposure DetailsModerate
Teriflunomide Dofetilide Tikosyn Increased dofetilide exposure Details Teriflunomide Encorafenib Braftovi Increased BCRP substrate exposure and an increased risk of BCRP substrate-related toxicities Details Teriflunomide Hydrocortisone Ala-Cort Increased hydrocortisone exposure and an increased risk of hydrocortisone-related adverse reactions Details Teriflunomide Hydrocortisone Injection A-Hydrocort® Increased hydrocortisone exposure and an increased risk of hydrocortisone-related adverse reactions Details Teriflunomide Levonorgestrel After banger Increased levonorgestrel exposure Details Teriflunomide Levonorgestrel Intrauterine System Kyleena Increased levonorgestrel exposure DetailsNo interactions on this page match that filter — try the next page or clear the filter.
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