Cabergoline

71 interactions 1 explained in plain English 69 cited references
Also sold as: Dostinex®
About Cabergoline

Cabergoline is used to treat hyperprolactinemia (high levels of prolactin, a natural substance that helps breast-feeding women produce milk but can cause symptoms such as infertility, sexual problems, and bone loss in women who are not breast-feeding or men). Cabergoline is in a class of medications called dopamine rec… Read the full Cabergoline drug information page →

Dr. Brian Staiger, PharmD, BCPS
Medically reviewed by Dr. Brian Staiger, PharmD, BCPS · Updated Jul 12, 2026 · Editorial policy · Data sources

Sources: FDA prescribing information (Structured Product Labeling), the published literature cited in each entry, DDInter 2.0 (a major open-access drug-interaction database), and legacy DrugBank interaction data distributed by the NIH's RxNav service (decommissioned in 2024) — analyzed and reviewed by our pharmacist team. How we build this library →

Major

Cabergoline Amisulpride Injection Barhemsys Reduced efficacy of cabergoline and reduced efficacy of dopamine-2 receptors Details Cabergoline Aripiprazole Injection Abilify Reduced efficacy of cabergoline and reduced efficacy of dopamine-2 receptors Details Cabergoline Asenapine Transdermal Patch Secuado Reduced efficacy of cabergoline and reduced efficacy of dopamine-2 receptors Details Cabergoline Acetophenazine Reduced efficacy of cabergoline and reduced efficacy of dopamine-2 receptors Details Cabergoline Alizapride Reduced efficacy of cabergoline and reduced efficacy of dopamine-2 receptors Details Cabergoline Amisulpride Barhemsys Reduced efficacy of cabergoline and reduced efficacy of dopamine-2 receptors Details Cabergoline Aripiprazole Abilify Reduced efficacy of cabergoline and reduced efficacy of dopamine-2 receptors Details Cabergoline Aripiprazole Lauroxil Aristada Reduced efficacy of cabergoline and reduced efficacy of dopamine-2 receptors Details Cabergoline Asenapine Saphris Reduced efficacy of cabergoline and reduced efficacy of dopamine-2 receptors Details Cabergoline Benperidol Reduced efficacy of cabergoline and reduced efficacy of dopamine-2 receptors Details Cabergoline Brexpiprazole Rexulti Reduced efficacy of cabergoline and reduced efficacy of dopamine-2 receptors Details Cabergoline Bromopride Reduced efficacy of cabergoline and reduced efficacy of dopamine-2 receptors Details Cabergoline Bromperidol Reduced efficacy of cabergoline and reduced efficacy of dopamine-2 receptors Details Cabergoline Cariprazine Vraylar Explained Reduced efficacy of cabergoline and reduced efficacy of dopamine-2 receptors Details Cabergoline Chlorpromazine Reduced efficacy of cabergoline and reduced efficacy of dopamine-2 receptors Details Cabergoline Chlorprothixene Reduced efficacy of cabergoline and reduced efficacy of dopamine-2 receptors Details Cabergoline Clozapine Clozaril Reduced efficacy of cabergoline and reduced efficacy of dopamine-2 receptors Details Cabergoline Dixyrazine Reduced efficacy of cabergoline and reduced efficacy of dopamine-2 receptors Details Cabergoline Domperidone Reduced efficacy of cabergoline and reduced efficacy of dopamine-2 receptors Details Cabergoline Droperidol Reduced efficacy of cabergoline and reduced efficacy of dopamine-2 receptors Details Cabergoline Ethopropazine Reduced efficacy of cabergoline and reduced efficacy of dopamine-2 receptors Details Cabergoline Fexofenadine Allegra Reduced efficacy of cabergoline and reduced efficacy of dopamine-2 receptors Details Cabergoline Flupenthixol Reduced efficacy of cabergoline and reduced efficacy of dopamine-2 receptors Details Cabergoline Fluphenazine Reduced efficacy of cabergoline and reduced efficacy of dopamine-2 receptors Details Cabergoline Fluspirilene Reduced efficacy of cabergoline and reduced efficacy of dopamine-2 receptors Details Cabergoline Haloperidol Loss of antiparkinson efficacy Details Cabergoline Iloperidone Fanapt Reduced efficacy of cabergoline and reduced efficacy of dopamine-2 receptors Details Cabergoline Itraconazole Sporanox Increased cabergoline exposure and an increased risk of cabergoline-related adverse effects Details Cabergoline Loxapine Adasuve Reduced efficacy of cabergoline and reduced efficacy of dopamine-2 receptors Details Cabergoline Lumateperone Caplyta Reduced efficacy of cabergoline and reduced efficacy of dopamine-2 receptors Details Cabergoline Lurasidone Latuda Reduced efficacy of cabergoline and reduced efficacy of dopamine-2 receptors Details Cabergoline Mesoridazine Reduced efficacy of cabergoline and reduced efficacy of dopamine-2 receptors Details Cabergoline Methdilazine Reduced efficacy of cabergoline and reduced efficacy of dopamine-2 receptors Details Cabergoline Methotrimeprazine Reduced efficacy of cabergoline and reduced efficacy of dopamine-2 receptors Details Cabergoline Metoclopramide Diminished effectiveness of metoclopramide and the dopaminergic agent Details Cabergoline Metopimazine Reduced efficacy of cabergoline and reduced efficacy of dopamine-2 receptors Details Cabergoline Molindone Reduced efficacy of cabergoline and reduced efficacy of dopamine-2 receptors Details Cabergoline Olanzapine Reduced efficacy of dopamine agonist Details Cabergoline Paliperidone Erzofri Reduced efficacy of cabergoline and reduced efficacy of dopamine-2 receptors Details

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Educational information only, not medical advice. Always confirm interactions with your pharmacist or prescriber before making any change to your medications.