Rosuvastatin

24 interactions 2 explained in plain English
Also sold as: Crestor Crestor® Ezallor Ezallor®
About Rosuvastatin

Rosuvastatin is a statin used to lower cholesterol and reduce the risk of heart attack and stroke. Read the full Rosuvastatin drug information page →

Dr. Brian Staiger, PharmD, BCPS
Medically reviewed by Dr. Brian Staiger, PharmD, BCPS · Updated Jun 30, 2026 · Editorial policy · Data sources

Sources: FDA prescribing information (Structured Product Labeling), the published literature cited in each entry, DDInter 2.0 (a major open-access drug-interaction database), and legacy DrugBank interaction data distributed by the NIH's RxNav service (decommissioned in 2024) — analyzed and reviewed by our pharmacist team. How we build this library →

Major

Rosuvastatin Colchicine Colcrys Explained An increased risk of myopathy or rhabdomyolysis Details Rosuvastatin Asciminib Scemblix Increased rosuvastatin exposure and an increased risk of rosuvastatin-related adverse effects Details Rosuvastatin Belumosudil Rezurock Explained Increased rosuvastatin exposure and an increased risk of myopathy and rhabdomyolysis Details Rosuvastatin Abiraterone Abirtega Increased rosuvastatin exposure and increased risk of myopathy Details Rosuvastatin Capmatinib Tabrecta Increased rosuvastatin exposure and an increased risk of myopathy and rhabdomyolysis Details Rosuvastatin Cyclosporine Injection Atopica Increased rosuvastatin exposure and an increased risk of myopathy and rhabdomyolysis Details Rosuvastatin Cyclosporine Ophthalmic Cequa Increased rosuvastatin exposure and an increased risk of myopathy and rhabdomyolysis Details Rosuvastatin Daptomycin Cubicin Increased risk of myopathy or rhabdomyolysis Details Rosuvastatin Daptomycin Injection Cubicin Increased risk of myopathy or rhabdomyolysis Details Rosuvastatin Darolutamide Nubeqa Increased rosuvastatin exposure and an increased risk of myopathy and rhabdomyolysis Details Rosuvastatin Elacestrant Orserdu Increased rosuvastatin exposure and an increased risk of rosuvastatin-related adverse effects Details Rosuvastatin Eluxadoline Viberzi Increased rosuvastatin exposure Details Rosuvastatin Enasidenib Idhifa Increased rosuvastatin exposure and an increased risk of myopathy and rhabdomyolysis Details Rosuvastatin Febuxostat Uloric Increased rosuvastatin exposure and an increased risk of myopathy and rhabdomyolysis Details Rosuvastatin Fostamatinib Tavalisse Increased rosuvastatin exposure and an increased risk of myopathy and rhabdomyolysis Details Rosuvastatin Gemfibrozil Lopid Increased rosuvastatin exposure and an increased risk of myopathy and rhabdomyolysis Details Rosuvastatin Leflunomide Arava Increased rosuvastatin exposure and an increased risk of myopathy and rhabdomyolysis Details Rosuvastatin Leniolisib Joenja Increased BCRP/OATP1B1/OATP1B3 substrate exposure Details Rosuvastatin Letermovir Injection Prevymis Increased statins exposure and an increased risk for myopathy and rhabdomyolysis Details Rosuvastatin Midostaurin Rydapt Increased BCRP and OATP1B1 substrate exposure Details Rosuvastatin Niacin Endur-Acin An increased risk of myopathy or rhabdomyolysis Details

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Educational information only, not medical advice. Always confirm interactions with your pharmacist or prescriber before making any change to your medications.